Synthesis of Aryl-Substituted 1,4-Dihydroquinolines by [4+2] Cycloaddition of Benzyne with 1-Azadienes

Abstract The synthesis of aryl-substituted 1,4-dihydroquinolines can be achieved using a [4+2] cycloaddition between benzyne and various aryl-substituted 1-azadienes. The conditions are tolerated by N-aryl-, alkyl-, tosyl-, and TERT-butoxycarbonyl-protected 1-azadienes. A short synthesis of the fung...

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Bibliographic Details

Published in:	Synlett 2012-02, Vol.2012 (3), p.389-392
Main Authors:	Stokes, Sean, Bekkam, Markondaiah, Rupp, Madeline, Mead, Keith T.
Format:	Article
Language:	English
Subjects:	Chemistry Exact sciences and technology Heterocyclic compounds Heterocyclic compounds with only one n hetero atom and condensed derivatives letter Organic chemistry Preparations and properties
Citations:	Items that cite this one
Online Access:	Get full text
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