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The influence of drug distribution and drug-target binding on target occupancy: The rate-limiting step approximation
by
de Witte, W.E.A.
,
Vauquelin, G.
,
van der Graaf, P.H.
,
de Lange, E.C.M.
Published in
European journal of pharmaceutical sciences
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European Journal Of Pharmaceutical Sciences
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Binding Kinetics
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Diffusion
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Distribution
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Drug Delivery Systems
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Humans
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Kinetics
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Life Sciences & Biomedicine
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Pharmaceutical Preparations - Administration & Dosage
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Pharmaceutical Preparations - Metabolism
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Pharmacokinetics
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Pharmacology & Pharmacy
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Rate-Limiting Step
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Rebinding
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Science & Technology
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Tissue Distribution - Drug Effects
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