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Search Results - Zrada, Matthew M
Search Results - Zrada, Matthew M
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The anesthetized guinea pig: An effective early cardiovascular derisking and lead optimization model
by
Morissette, Pierre
,
Nishida, Masahiro
,
Trepakova, Elena
,
Imredy, John
,
Lagrutta, Armando
,
Chaves, Alysia
,
Hoagland, Kimberly
,
Hoe, Chao-Min Lei
,
Zrada, Matthew M.
,
Travis, Jeffrey J.
,
Zingaro, Gloria J.
,
Gerenser, Pamela
,
Friedrichs, Greg
,
Salata, Joseph J.
Published in
Journal of pharmacological and toxicological methods
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Discovery of 1,4-Substituted Piperidines as Potent and Selective Inhibitors of T-Type Calcium Channels
by
Yang, Zhi-Qiang
,
Barrow, James C
,
Shipe, William D
,
Schlegel, Kelly-Ann S
,
Shu, Youheng
,
Yang, F. Vivien
,
Lindsley, Craig W
,
Rittle, Kenneth E
,
Bock, Mark G
,
Hartman, George D
,
Uebele, Victor N
,
Nuss, Cindy E
,
Fox, Steve V
,
Kraus, Richard L
,
Doran, Scott M
,
Connolly, Thomas M
,
Tang, Cuyue
,
Ballard, Jeanine E
,
Kuo, Yuhsin
,
Adarayan, Emily D
,
Prueksaritanont, Thomayant
,
Zrada, Matthew M
,
Marino, Michael J
,
Graufelds, Valerie Kuzmick
,
DiLella, Anthony G
,
Reynolds, Ian J
,
Vargas, Hugo M
,
Bunting, Patricia B
,
Woltmann, Richard F
,
Magee, Michael M
,
Koblan, Kenneth S
,
Renger, John J
Published in
Journal of medicinal chemistry
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MK-8825: A potent and selective CGRP receptor antagonist with good oral activity in rats
by
Bell, Ian M.
,
Stump, Craig A.
,
Gallicchio, Steven N.
,
Staas, Donnette D.
,
Zartman, C. Blair
,
Moore, Eric L.
,
Sain, Nova
,
Urban, Mark
,
Bruno, Joseph G.
,
Calamari, Amy
,
Kemmerer, Amanda L.
,
Mosser, Scott D.
,
Fandozzi, Christine
,
White, Rebecca B.
,
Zrada, Matthew M.
,
Selnick, Harold G.
,
Graham, Samuel L.
,
Vacca, Joseph P.
,
Kane, Stefanie A.
,
Salvatore, Christopher A.
Published in
Bioorganic & medicinal chemistry letters
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Kinesin spindle protein (KSP) inhibitors. Part V: Discovery of 2-propylamino-2,4-diaryl-2,5-dihydropyrroles as potent, water-soluble KSP inhibitors, and modulation of their basicit...
by
Cox, Christopher D.
,
Breslin, Michael J.
,
Whitman, David B.
,
Coleman, Paul J.
,
Garbaccio, Robert M.
,
Fraley, Mark E.
,
Zrada, Matthew M.
,
Buser, Carolyn A.
,
Walsh, Eileen S.
,
Hamilton, Kelly
,
Lobell, Robert B.
,
Tao, Weikang
,
Abrams, Marc T.
,
South, Vicki J.
,
Huber, Hans E.
,
Kohl, Nancy E.
,
Hartman, George D.
Published in
Bioorganic & medicinal chemistry letters
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8-Hydroxy-3,4-dihydropyrrolo[1,2- a]pyrazine-1(2 H)-one HIV-1 integrase inhibitors
by
Fisher, Thorsten E.
,
Kim, Boyoung
,
Staas, Donnette D.
,
Lyle, Terry A.
,
Young, Steven D.
,
Vacca, Joseph P.
,
Zrada, Matthew M.
,
Hazuda, Daria J.
,
Felock, Peter J.
,
Schleif, William A.
,
Gabryelski, Lori J.
,
Anari, M. Reza
,
Kochansky, Christopher J.
,
Wai, John S.
Published in
Bioorganic & medicinal chemistry
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A potent and orally active HIV-1 integrase inhibitor
by
Egbertson, Melissa S.
,
Moritz, H. Marie
,
Melamed, Jeffrey Y.
,
Han, Wei
,
Perlow, Debra S.
,
Kuo, Michelle S.
,
Embrey, Mark
,
Vacca, Joseph P.
,
Zrada, Matthew M.
,
Cortes, Amanda R.
,
Wallace, Audrey
,
Leonard, Yvonne
,
Hazuda, Daria J.
,
Miller, Michael D.
,
Felock, Peter J.
,
Stillmock, Kara A.
,
Witmer, Marc V.
,
Schleif, William
,
Gabryelski, Lori J.
,
Moyer, Gregory
,
Ellis, Joan D.
,
Jin, Lixia
,
Xu, Wei
,
Braun, Matthew P.
,
Kassahun, Kellem
,
Tsou, Nancy N.
,
Young, Steven D.
Published in
Bioorganic & medicinal chemistry letters
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9-Hydroxyazafluorenes and Their Use in Thrombin Inhibitors
by
Stauffer, Kenneth J
,
Williams, Peter D
,
Selnick, Harold G
,
Nantermet, Philippe G
,
Newton, Christina L
,
Homnick, Carl F
,
Zrada, Matthew M
,
Lewis, S. Dale
,
Lucas, Bobby J
,
Krueger, Julie A
,
Pietrak, Beth L
,
Lyle, Elizabeth A
,
Singh, Rominder
,
Miller-Stein, Cynthia
,
White, Rebecca B
,
Wong, Bradley
,
Wallace, Audrey A
,
Sitko, Gary R
,
Cook, Jacquelyn J
,
Holahan, Marie A
,
Stranieri-Michener, Maria
,
Leonard, Yvonne M
,
Lynch, Joseph J
,
McMasters, Daniel R
,
Yan, Youwei
Published in
Journal of medicinal chemistry
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Design, Synthesis, and Evaluation of a Novel 4-Aminomethyl-4-fluoropiperidine as a T-Type Ca2+ Channel Antagonist
by
Shipe, William D
,
Barrow, James C
,
Yang, Zhi-Qiang
,
Lindsley, Craig W
,
Yang, F. Vivien
,
Schlegel, Kelly-Ann S
,
Shu, Youheng
,
Rittle, Kenneth E
,
Bock, Mark G
,
Hartman, George D
,
Tang, Cuyue
,
Ballard, Jeanine E
,
Kuo, Yuhsin
,
Adarayan, Emily D
,
Prueksaritanont, Thomayant
,
Zrada, Matthew M
,
Uebele, Victor N
,
Nuss, Cindy E
,
Connolly, Thomas M
,
Doran, Scott M
,
Fox, Steven V
,
Kraus, Richard L
,
Marino, Michael J
,
Graufelds, Valerie Kuzmick
,
Vargas, Hugo M
,
Bunting, Patricia B
,
Hasbun-Manning, Martha
,
Evans, Rose M
,
Koblan, Kenneth S
,
Renger, John J
Published in
Journal of medicinal chemistry
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Development of an efficient and selective radioligand for bradykinin B1 receptor occupancy studies
by
SU, Dai-Shi
,
MARKOWITZ, M. Kristine
,
WALLACE, Michael A
,
RAAB, Conrad E
,
DEAN, Dennis C
,
PETTIBONE, Douglas J
,
FREIDINGER, Roger M
,
BOCK, Mark G
,
MURPHY, Kathy L
,
WAN, Bang-Lin
,
ZRADA, Matthew M
,
HARRELL, C. Meacham
,
O'MALLEY, Stacy S
,
HESS, J. Fred
,
RANSOM, Rick W
,
CHANG, Ray S
Published in
Bioorganic & medicinal chemistry letters
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Development of an efficient and selective radioligand for bradykinin B 1 receptor occupancy studies
by
Su, Dai-Shi
,
Markowitz, M. Kristine
,
Murphy, Kathy L.
,
Wan, Bang-Lin
,
Zrada, Matthew M.
,
Harrell, C. Meacham
,
O’Malley, Stacy S.
,
Hess, J. Fred
,
Ransom, Rick W.
,
Chang, Ray S.
,
Wallace, Michael A.
,
Raab, Conrad E.
,
Dean, Dennis C.
,
Pettibone, Douglas J.
,
Freidinger, Roger M.
,
Bock, Mark G.
Published in
Bioorganic & medicinal chemistry letters
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Design, Synthesis, and Evaluation of a Novel 4-Aminomethyl-4-fluoropiperidine as a T-Type Ca 2+ Channel Antagonist
by
Shipe, William D.
,
Barrow, James C.
,
Yang, Zhi-Qiang
,
Lindsley, Craig W.
,
Yang, F. Vivien
,
Schlegel, Kelly-Ann S.
,
Shu, Youheng
,
Rittle, Kenneth E.
,
Bock, Mark G.
,
Hartman, George D.
,
Tang, Cuyue
,
Ballard, Jeanine E.
,
Kuo, Yuhsin
,
Adarayan, Emily D.
,
Prueksaritanont, Thomayant
,
Zrada, Matthew M.
,
Uebele, Victor N.
,
Nuss, Cindy E.
,
Connolly, Thomas M.
,
Doran, Scott M.
,
Fox, Steven V.
,
Kraus, Richard L.
,
Marino, Michael J.
,
Graufelds, Valerie Kuzmick
,
Vargas, Hugo M.
,
Bunting, Patricia B.
,
Hasbun-Manning, Martha
,
Evans, Rose M.
,
Koblan, Kenneth S.
,
Renger, John J.
Published in
Journal of medicinal chemistry
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Structure-affinity relationships of arylquinolizines at .alpha.-adrenoceptors
by
Huff, Joel R
,
Baldwin, John J
,
DeSolms, S. Jane
,
Guare, James P
,
Hunt, Cecilia A
,
Randall, William C
,
Sanders, William S
,
Smith, Steven J
,
Vacca, Joseph P
,
Zrada, Matthew M
Published in
Journal of medicinal chemistry
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