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Quantifying the chameleonic properties of macrocycles and other high-molecular-weight drugs
by
Whitty, Adrian
,
Zhong, Mengqi
,
Viarengo, Lauren
,
Beglov, Dmitri
,
Hall, David R.
,
Vajda, Sandor
Published in
Drug discovery today
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Conformational Effects on the Passive Membrane Permeability of Synthetic Macrocycles
by
Rzepiela, Anna A.
,
Viarengo-Baker, Lauren A.
,
Tatarskii, Victor
,
Kombarov, Roman
,
Whitty, Adrian
Published in
Journal of medicinal chemistry
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Defining and navigating macrocycle chemical space
by
Viarengo-Baker, Lauren A
,
Brown, Lauren E
,
Rzepiela, Anna A
,
Whitty, Adrian
Published in
Chemical science (Cambridge)
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Recapitulating the Binding Affinity of Nrf2 for KEAP1 in a Cyclic Heptapeptide, Guided by NMR, X‑ray Crystallography, and Machine Learning
by
Ortet, Paula C
,
Muellers, Samantha N
,
Viarengo-Baker, Lauren A
,
Streu, Kristina
,
Szymczyna, Blair R
,
Beeler, Aaron B
,
Allen, Karen N
,
Whitty, Adrian
Published in
Journal of the American Chemical Society
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