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Bipartite interface of the measles virus phosphoprotein X domain with the large polymerase protein regulates viral polymerase dynamics
by
Du Pont, Venice
,
Jiang, Yi
,
Plemper, Richard K
Published in
PLoS pathogens
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The Nucleoside/Nucleotide Analogs Tenofovir and Emtricitabine Are Inactive against SARS-CoV-2
by
Feng, Joy Y.
,
Du Pont, Venice
,
Babusis, Darius
,
Gordon, Calvin J.
,
Tchesnokov, Egor P.
,
Perry, Jason K.
,
Duong, Vincent
,
Vijjapurapu, Arya
,
Zhao, Xiaofeng
,
Chan, Julie
,
Cohen, Cal
,
Juneja, Kavita
,
Cihlar, Tomas
,
Götte, Matthias
,
Bilello, John P.
Published in
Molecules (Basel, Switzerland)
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Remdesivir Inhibits SARS-CoV-2 in Human Lung Cells and Chimeric SARS-CoV Expressing the SARS-CoV-2 RNA Polymerase in Mice
by
Pruijssers, Andrea J.
,
George, Amelia S.
,
Schäfer, Alexandra
,
Leist, Sarah R.
,
Gralinksi, Lisa E.
,
Dinnon, Kenneth H.
,
Yount, Boyd L.
,
Agostini, Maria L.
,
Stevens, Laura J.
,
Chappell, James D.
,
Lu, Xiaotao
,
Hughes, Tia M.
,
Gully, Kendra
,
Martinez, David R.
,
Brown, Ariane J.
,
Graham, Rachel L.
,
Perry, Jason K.
,
Du Pont, Venice
,
Pitts, Jared
,
Ma, Bin
,
Babusis, Darius
,
Murakami, Eisuke
,
Feng, Joy Y.
,
Bilello, John P.
,
Porter, Danielle P.
,
Cihlar, Tomas
,
Baric, Ralph S.
,
Denison, Mark R.
,
Sheahan, Timothy P.
Published in
Cell Reports
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Remdesivir and GS-441524 Retain Antiviral Activity against Delta, Omicron, and Other Emergent SARS-CoV-2 Variants
by
Pitts, Jared
,
Li, Jiani
,
Perry, Jason K
,
Du Pont, Venice
,
Riola, Nicholas
,
Rodriguez, Lauren
,
Lu, Xianghan
,
Kurhade, Chaitanya
,
Xie, Xuping
,
Camus, Gregory
,
Manhas, Savrina
,
Martin, Ross
,
Shi, Pei-Yong
,
Cihlar, Tomas
,
Porter, Danielle P
,
Mo, Hongmei
,
Maiorova, Evguenia
,
Bilello, John P
Published in
Antimicrobial agents and chemotherapy
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In Vitro Selection of Remdesivir-Resistant SARS-CoV-2 Demonstrates High Barrier to Resistance
by
Checkmahomed, Liva
,
Carbonneau, Julie
,
Du Pont, Venice
,
Riola, Nicholas C
,
Perry, Jason K
,
Li, Jiani
,
Paré, Bastien
,
Simpson, Shawn M
,
Smith, Martin A
,
Porter, Danielle P
,
Boivin, Guy
Published in
Antimicrobial agents and chemotherapy
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Status of antiviral therapeutics against rabies virus and related emerging lyssaviruses
by
Du Pont, Venice
,
Plemper, Richard K
,
Schnell, Matthias J
Published in
Current opinion in virology
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Identification and Characterization of a Small-Molecule Rabies Virus Entry Inhibitor
by
Du Pont, Venice
,
Wirblich, Christoph
,
Yoon, Jeong-Joong
,
Cox, Robert M
,
Schnell, Matthias J
,
Plemper, Richard K
Published in
Journal of virology
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Prodrugs of a 1′-CN-4-Aza-7,9-dideazaadenosine C‑Nucleoside Leading to the Discovery of Remdesivir (GS-5734) as a Potent Inhibitor of Respiratory Syncytial Virus with Efficacy in t...
by
Mackman, Richard L
,
Hui, Hon C
,
Perron, Michel
,
Murakami, Eisuke
,
Palmiotti, Christopher
,
Lee, Gary
,
Stray, Kirsten
,
Zhang, Lijun
,
Goyal, Bindu
,
Chun, Kwon
,
Byun, Daniel
,
Siegel, Dustin
,
Simonovich, Scott
,
Du Pont, Venice
,
Pitts, Jared
,
Babusis, Darius
,
Vijjapurapu, Arya
,
Lu, Xianghan
,
Kim, Cynthia
,
Zhao, Xiaofeng
,
Chan, Julie
,
Ma, Bin
,
Lye, Diane
,
Vandersteen, Adelle
,
Wortman, Sarah
,
Barrett, Kimberly T
,
Toteva, Maria
,
Jordan, Robert
,
Subramanian, Raju
,
Bilello, John P
,
Cihlar, Tomas
Published in
Journal of medicinal chemistry
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Discovery of GS-5245 (Obeldesivir), an Oral Prodrug of Nucleoside GS-441524 That Exhibits Antiviral Efficacy in SARS-CoV-2-Infected African Green Monkeys
by
Mackman, Richard L.
,
Kalla, Rao V.
,
Babusis, Darius
,
Pitts, Jared
,
Barrett, Kimberly T.
,
Chun, Kwon
,
Du Pont, Venice
,
Rodriguez, Lauren
,
Moshiri, Jasmine
,
Xu, Yili
,
Lee, Michael
,
Lee, Gary
,
Bleier, Blake
,
Nguyen, Anh-Quan
,
O’Keefe, B. Michael
,
Ambrosi, Andrea
,
Cook, Meredith
,
Yu, Joy
,
Dempah, Kassibla Elodie
,
Bunyan, Elaine
,
Riola, Nicholas C.
,
Lu, Xianghan
,
Liu, Renmeng
,
Davie, Ashley
,
Hsiang, Tien-Ying
,
Dearing, Justin
,
Vermillion, Meghan
,
Gale, Michael
,
Niedziela-Majka, Anita
,
Feng, Joy Y.
,
Hedskog, Charlotte
,
Bilello, John P.
,
Subramanian, Raju
,
Cihlar, Tomas
Published in
Journal of medicinal chemistry
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539. Efficacy in Multiple SARS-CoV-2 Animal Models Supports Phase 3 Dose Selection for Obeldesivir
by
Pitts, Jared
,
Babusis, Darius
,
Humeniuk, Rita
,
Martinez, David
,
Cox, Robert M
,
Schäfer, Alexandra
,
Riola, Nicholas C
,
Feng, Joy
,
Du Pont, Venice
,
Anoshchenko, Olena
,
Vermillion, Meghan
,
Abdelghany, Mazin
,
Hyland, Robert H
,
Girish, Sandhya
,
Sheahan, Timothy P
,
Plemper, Richard K
,
Baric, Ralph S
,
Cihlar, Tomas
,
Llewellyn, Joe
,
Winter, Helen
,
Bannister, Roy
,
Subramanian, Raju
,
Mackman, Richard L
,
Bilello, John P
Published in
Open forum infectious diseases
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Therapeutic efficacy of an oral nucleoside analog of remdesivir against SARS-CoV-2 pathogenesis in mice
by
Schafer, Alexandra
,
Martinez, David R
,
Won, John J
,
Moreira, Fernanado R
,
Brown, Ariane J
,
Gully, Kendra L
,
Kalla, Rao
,
Kwon Chun
,
Venice Du Pont
,
Babusis, Darius
,
Tang, Jennifer
,
Murakami, Eisuke
,
Subramanian, Raju
,
Barrett, Kimberly T
,
Bleier, Blake J
,
Bannister, Roy
,
Feng, Joy Y
,
Bilello, John P
,
Cihlar, Tomas
,
Mackman, Richard L
,
Montgomery, Stephanie A
,
Baric, Ralph S
,
Sheahan, Timothy P
Published in
bioRxiv
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In Vitro Selection of Remdesivir-Resistant SARS-CoV-2 Demonstrates High Barrier to Resistance
by
Checkmahomed, Liva
,
Venice Du Pont
,
Riola, Nicholas C
,
Perry, Jason
,
Li, Jiani
,
Danielle Poulin Porter
,
Boivin, Guy
Published in
bioRxiv
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Remdesivir and GS-441524 retain antiviral activity against Delta, Omicron, and other emergent SARS-CoV-2 variants
by
Pitts, Jared
,
Li, Jiani
,
Perry, Jason
,
Venice Du Pont
,
Riola, Nicholas
,
Rodriguez, Lauren
,
Lu, Xianghan
,
Kurhade, Chaitanya
,
Xie, Xuping
,
Camus, Gregory
,
Manhas, Savrina
,
Ross, Martin
,
Pei-Yong, Shi
,
Cihlar, Tomas
,
Danielle Poulin Porter
,
Mo, Hongmei
,
Maiorova, Evguenia S
,
Bilello, John P
Published in
bioRxiv
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