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Small Molecule Tools to Study Cellular Target Engagement for the Intracellular Allosteric Binding Site of GPCRs
by
Huber, Max E.
,
Toy, Lara
,
Schmidt, Maximilian F.
,
Weikert, Dorothee
,
Schiedel, Matthias
Published in
Chemistry : a European journal
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Fluorescent Ligands Targeting the Intracellular Allosteric Binding Site of the Chemokine Receptor CCR2
by
Toy, Lara
,
Huber, Max E.
,
Schmidt, Maximilian F.
,
Weikert, Dorothee
,
Schiedel, Matthias
Published in
ACS chemical biology
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A Chemical Biology Toolbox Targeting the Intracellular Binding Site of CCR9: Fluorescent Ligands, New Drug Leads and PROTACs
by
Huber, Max E.
,
Toy, Lara
,
Schmidt, Maximilian F.
,
Vogt, Hannah
,
Budzinski, Julian
,
Wiefhoff, Martin F. J.
,
Merten, Nicole
,
Kostenis, Evi
,
Weikert, Dorothee
,
Schiedel, Matthias
Published in
Angewandte Chemie International Edition
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Frontispiece: Small Molecule Tools to Study Cellular Target Engagement for the Intracellular Allosteric Binding Site of GPCRs
by
Huber, Max E.
,
Toy, Lara
,
Schmidt, Maximilian F.
,
Weikert, Dorothee
,
Schiedel, Matthias
Published in
Chemistry : a European journal
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Fluorescent Ligands Enable Target Engagement Studies for the Intracellular Allosteric Binding Site of the Chemokine Receptor CXCR2
by
Huber, Max E.
,
Wurnig, Silas
,
Toy, Lara
,
Weiler, Corinna
,
Merten, Nicole
,
Kostenis, Evi
,
Hansen, Finn K.
,
Schiedel, Matthias
Published in
Journal of medicinal chemistry
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Development of First-in-Class Dual Sirt2/HDAC6 Inhibitors as Molecular Tools for Dual Inhibition of Tubulin Deacetylation
by
Sinatra, Laura
,
Vogelmann, Anja
,
Friedrich, Florian
,
Tararina, Margarita A.
,
Neuwirt, Emilia
,
Colcerasa, Arianna
,
König, Philipp
,
Toy, Lara
,
Yesiloglu, Talha Z.
,
Hilscher, Sebastian
,
Gaitzsch, Lena
,
Papenkordt, Niklas
,
Zhai, Shiyang
,
Zhang, Lin
,
Romier, Christophe
,
Einsle, Oliver
,
Sippl, Wolfgang
,
Schutkowski, Mike
,
Gross, Olaf
,
Bendas, Gerd
,
Christianson, David W.
,
Hansen, Finn K.
,
Jung, Manfred
,
Schiedel, Matthias
Published in
Journal of medicinal chemistry
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Development of a NanoBRET Assay Platform to Detect Intracellular Ligands for the Chemokine Receptors CCR6 and CXCR1
by
Huber, Max E.
,
Wurnig, Silas L.
,
Moumbock, Aurélien F. A.
,
Toy, Lara
,
Kostenis, Evi
,
Alonso Bartolomé, Ana
,
Szpakowska, Martyna
,
Chevigné, Andy
,
Günther, Stefan
,
Hansen, Finn K.
,
Schiedel, Matthias
Published in
ChemMedChem
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Fluorophore-Labeled Pyrrolones Targeting the Intracellular Allosteric Binding Site of the Chemokine Receptor CCR1
by
Toy, Lara
,
Huber, Max E.
,
Lee, Minhee
,
Bartolomé, Ana Alonso
,
Ortiz Zacarías, Natalia V.
,
Nasser, Sherif
,
Scholl, Stephan
,
Zlotos, Darius P.
,
Mandour, Yasmine M.
,
Heitman, Laura H.
,
Szpakowska, Martyna
,
Chevigné, Andy
,
Schiedel, Matthias
Published in
ACS pharmacology & translational science
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Chemisch‐biologischer Werkzeugkasten für die intrazelluläre Bindungsstelle von CCR9: Fluoreszierende Liganden, neue Leitstrukturen und PROTACs
by
Huber, Max E.
,
Toy, Lara
,
Schmidt, Maximilian F.
,
Vogt, Hannah
,
Budzinski, Julian
,
Wiefhoff, Martin F. J.
,
Merten, Nicole
,
Kostenis, Evi
,
Weikert, Dorothee
,
Schiedel, Matthias
Published in
Angewandte Chemie
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Chemisch‐biologischer Werkzeugkasten für die intrazelluläre Bindungsstelle von CCR9: Fluoreszierende Liganden, neue Leitstrukturen und PROTACs
by
Huber, Max E.
,
Toy, Lara
,
Schmidt, Maximilian F.
,
Vogt, Hannah
,
Budzinski, Julian
,
Wiefhoff, Martin F. J.
,
Merten, Nicole
,
Kostenis, Evi
,
Weikert, Dorothee
,
Schiedel, Matthias
Published in
Angewandte Chemie
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