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Search Results - Thabault, Léopold
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Rational Design of Original Fused-Cycle Selective Inhibitors of Tryptophan 2,3-Dioxygenase
by
Kozlova, Arina
,
Thabault, Léopold
,
Liberelle, Maxime
,
Klaessens, Simon
,
Prévost, Julien R. C
,
Mathieu, Caroline
,
Pilotte, Luc
,
Stroobant, Vincent
,
Van den Eynde, Benoît
,
Frédérick, Raphaël
Published in
Journal of medicinal chemistry
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Interrogating the Lactate Dehydrogenase Tetramerization Site Using (Stapled) Peptides
by
Thabault, Léopold
,
Brisson, Lucie
,
Brustenga, Chiara
,
Martinez Gache, Santiago A
,
Prévost, Julien R. C
,
Kozlova, Arina
,
Spillier, Quentin
,
Liberelle, Maxime
,
Benyahia, Zohra
,
Messens, Joris
,
Copetti, Tamara
,
Sonveaux, Pierre
,
Frédérick, Raphaël
Published in
Journal of medicinal chemistry
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Olaparib Is a Mitochondrial Complex I Inhibitor That Kills Temozolomide-Resistant Human Glioblastoma Cells
by
Zampieri, Luca X
,
Sboarina, Martina
,
Cacace, Andrea
,
Grasso, Debora
,
Thabault, Léopold
,
Hamelin, Loïc
,
Vazeille, Thibaut
,
Dumon, Elodie
,
Rossignol, Rodrigue
,
Frédérick, Raphaël
,
Sonveaux, Etienne
,
Lefranc, Florence
,
Sonveaux, Pierre
Published in
International journal of molecular sciences
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Correction to “Rational Design of Original Fused-Cycle Selective Inhibitors of Tryptophan 2,3-Dioxygenase”
by
Kozlova, Arina
,
Thabault, Léopold
,
Liberelle, Maxime
,
Klaessens, Simon
,
Prévost, Julien R. C
,
Mathieu, Caroline
,
Pilotte, Luc
,
Stroobant, Vincent
,
Van den Eynde, Benoît
,
Frédérick, Raphaël
Published in
Journal of medicinal chemistry
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Targeting protein self-association in drug design
by
Thabault, Léopold
,
Liberelle, Maxime
,
Frédérick, Raphaël
Published in
Drug discovery today
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Unravelling the Allosteric Targeting of PHGDH at the ACT-Binding Domain with a Photoactivatable Diazirine Probe and Mass Spectrometry Experiments
by
Spillier, Quentin
,
Ravez, Séverine
,
Dochain, Simon
,
Vertommen, Didier
,
Thabault, Léopold
,
Feron, Olivier
,
Frédérick, Raphaël
Published in
Molecules (Basel, Switzerland)
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Discovery of a novel lactate dehydrogenase tetramerization domain using epitope mapping and peptides
by
Thabault, Léopold
,
Liberelle, Maxime
,
Koruza, Katarina
,
Yildiz, Esra
,
Joudiou, Nicolas
,
Messens, Joris
,
Brisson, Lucie
,
Wouters, Johan
,
Sonveaux, Pierre
,
Frédérick, Raphaël
Published in
The Journal of biological chemistry
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Discovery of small molecules interacting at lactate dehydrogenases tetrameric interface using a biophysical screening cascade
by
Thabault, Léopold
,
Brustenga, Chiara
,
Savoyen, Perrine
,
Van Gysel, Mégane
,
Wouters, Johan
,
Sonveaux, Pierre
,
Frédérick, Raphaël
,
Liberelle, Maxime
Published in
European journal of medicinal chemistry
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Investigation of chalcogen bioisosteric replacement in a series of heterocyclic inhibitors of tryptophan 2,3-dioxygenase
by
Kozlova, Arina
,
Thabault, Léopold
,
Dauguet, Nicolas
,
Deskeuvre, Marine
,
Stroobant, Vincent
,
Pilotte, Luc
,
Liberelle, Maxime
,
Van den Eynde, Benoît
,
Frédérick, Raphaël
Published in
European journal of medicinal chemistry
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1-(2-Hydroxybenzoyl)-thiosemicarbazides are promising antimicrobial agents targeting d-alanine-d-alanine ligase in bacterio
by
Ameryckx, Alice
,
Thabault, Léopold
,
Pochet, Lionel
,
Leimanis, Serge
,
Poupaert, Jacques H.
,
Wouters, Johan
,
Joris, Bernard
,
Van Bambeke, Françoise
,
Frédérick, Raphaël
Published in
European journal of medicinal chemistry
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The putative Escherichia coli dehydrogenase YjhC metabolises two dehydrated forms of N-acetylneuraminate produced by some sialidases
by
Kentache, Takfarinas
,
Thabault, Léopold
,
Peracchi, Alessio
,
Frédérick, Raphaël
,
Bommer, Guido T
,
Van Schaftingen, Emile
Published in
Bioscience reports
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The metalloprotein YhcH is an anomerase providing N-acetylneuraminate aldolase with the open form of its substrate
by
Kentache, Takfarinas
,
Thabault, Leopold
,
Deumer, Gladys
,
Haufroid, Vincent
,
Frédérick, Raphaël
,
Linster, Carole L.
,
Peracchi, Alessio
,
Veiga-da-Cunha, Maria
,
Bommer, Guido T.
,
Van Schaftingen, Emile
Published in
The Journal of biological chemistry
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