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Search Results - TACHIBANA-KONDO, Yukako
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Enhanced Inhibition of ERK Signaling by a Novel Allosteric MEK Inhibitor, CH5126766, That Suppresses Feedback Reactivation of RAF Activity
by
ISHII, Nobuya
,
HARADA, Naoki
,
AOKI, Toshihiro
,
SHIMMA, Nobuo
,
ARISAWA, Mikio
,
SOWA, Yoshihiro
,
POULIKAKOS, Poulikos I
,
ROSEN, Neal
,
AOKI, Yuko
,
SAKAI, Toshiyuki
,
JOSEPH, Eric W
,
OHARA, Kazuhiro
,
MIURA, Takaaki
,
SAKAMOTO, Hiroshi
,
MATSUDA, Yutaka
,
TOMII, Yasushi
,
TACHIBANA-KONDO, Yukako
,
LIKURA, Hitoshi
Published in
Cancer research (Chicago, Ill.)
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Abstract 2729: FGFR genetic alterations as a potential predictor of the sensitivity to CH5183284/Debio 1347, a selective FGFR inhibitor with a novel chemical scaffold
by
Nakanishi, Yoshito
,
Akiyama, Nukinori
,
Tsukaguchi, Toshiyuki
,
Tachibana-Kondo, Yukako
,
Fujii, Toshihiko
,
Sakata, Kiyoaki
,
Sase, Hitoshi
,
Isobe, Takehito
,
Sato, Yasuko
,
Morikami, Kenji
,
Shindoh, Hidetoshi
,
Mio, Toshiyuki
,
Ebiike, Hirosato
,
Taka, Naoki
,
Aoki, Yuko
,
Ishii, Nobuya
Published in
Cancer research (Chicago, Ill.)
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Abstract 3606: CH5126766 is a novel allosteric inhibitor of MEK that prevents its phosphorylation by RAF
by
Ishii, Nobuya
,
Harada, Naoki
,
Sakamoto, Hiroshi
,
Matsuda, Yutaka
,
Tomii, Yasushi
,
Tachibana-Kondo, Yukako
,
Miura, Takaaki
,
Ohara, Kazuhiro
,
Iikura, Hitoshi
,
Aoki, Toshihiro
,
Shimma, Nobuo
,
Arisawa, Mikio
,
Joseph, Eric
,
Poulikakos, Poulikos
,
Sowa, Yoshihiro
,
Rosen, Neal
,
Aoki, Yuko
,
Sakai, Toshiyuki
Published in
Cancer research (Chicago, Ill.)
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Cancer Research
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Allosteric Regulation
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Animals
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Antineoplastic Agents
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Antineoplastic Agents - Pharmacology
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Biological And Medical Sciences
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Cell Line, Tumor
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Coumarins - Pharmacology
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Enzyme Activation - Drug Effects
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Extracellular Signal-Regulated Map Kinases - Metabolism
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Feedback, Physiological - Drug Effects
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Female
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Humans
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Life Sciences & Biomedicine
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Map Kinase Kinase 1 - Antagonists & Inhibitors
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Map Kinase Kinase 1 - Chemistry
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Mice
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Mice, Inbred Balb C
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