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Search Results - Suresh, Rudrapatna S
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Discovery of Pyrazolopyridones as a Novel Class of Noncovalent DprE1 Inhibitor with Potent Anti-Mycobacterial Activity
by
Panda, Manoranjan
,
Ramachandran, Sreekanth
,
Ramachandran, Vasanthi
,
Shirude, Pravin S
,
Humnabadkar, Vaishali
,
Nagalapur, Kavitha
,
Sharma, Sreevalli
,
Kaur, Parvinder
,
Guptha, Supreeth
,
Narayan, Ashwini
,
Mahadevaswamy, Jyothi
,
Ambady, Anisha
,
Hegde, Naina
,
Rudrapatna, Suresh S
,
Hosagrahara, Vinayak P
,
Sambandamurthy, Vasan K
,
Raichurkar, Anandkumar
Published in
Journal of medicinal chemistry
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Lead Optimization of 1,4-Azaindoles as Antimycobacterial Agents
by
Shirude, Pravin S
,
Shandil, Radha K
,
Manjunatha, M. R
,
Sadler, Claire
,
Panda, Manoranjan
,
Panduga, Vijender
,
Reddy, Jitendar
,
Saralaya, Ramanatha
,
Nanduri, Robert
,
Ambady, Anisha
,
Ravishankar, Sudha
,
Sambandamurthy, Vasan K
,
Humnabadkar, Vaishali
,
Jena, Lalit K
,
Suresh, Rudrapatna S
,
Srivastava, Abhishek
,
Prabhakar, K. R
,
Whiteaker, James
,
McLaughlin, Robert E
,
Sharma, Sreevalli
,
Cooper, Christopher B
,
Mdluli, Khisi
,
Butler, Scott
,
Iyer, Pravin S
,
Narayanan, Shridhar
,
Chatterji, Monalisa
Published in
Journal of medicinal chemistry
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Aminoazabenzimidazoles, a Novel Class of Orally Active Antimalarial Agents
by
Hameed P, Shahul
,
Chinnapattu, Murugan
,
Shanbag, Gajanan
,
Manjrekar, Praveena
,
Koushik, Krishna
,
Raichurkar, Anandkumar
,
Patil, Vikas
,
Jatheendranath, Sandesh
,
Rudrapatna, Suresh S
,
Barde, Shubhada P
,
Rautela, Nikhil
,
Awasthy, Disha
,
Morayya, Sapna
,
Narayan, Chandan
,
Kavanagh, Stefan
,
Saralaya, Ramanatha
,
Bharath, Sowmya
,
Viswanath, Pavithra
,
Mukherjee, Kakoli
,
Bandodkar, Balachandra
,
Srivastava, Abhishek
,
Panduga, Vijender
,
Reddy, Jitender
,
Prabhakar, K. R
,
Sinha, Achyut
,
Jiménez-Díaz, María Belén
,
Martínez, María Santos
,
Angulo-Barturen, Iñigo
,
Ferrer, Santiago
,
Sanz, Laura María
,
Gamo, Francisco Javier
,
Duffy, Sandra
,
Avery, Vicky M
,
Magistrado, Pamela A
,
Lukens, Amanda K
,
Wirth, Dyann F
,
Waterson, David
,
Balasubramanian, V
,
Iyer, Pravin S
,
Narayanan, Shridhar
,
Hosagrahara, Vinayak
,
Sambandamurthy, Vasan K
,
Ramachandran, Sreekanth
Published in
Journal of medicinal chemistry
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Discovery of Imidazo[1,2‑a]pyridine Ethers and Squaramides as Selective and Potent Inhibitors of Mycobacterial Adenosine Triphosphate (ATP) Synthesis
by
Tantry, Subramanyam J
,
Markad, Shankar D
,
Shinde, Vikas
,
Bhat, Jyothi
,
Balakrishnan, Gayathri
,
Gupta, Amit K
,
Ambady, Anisha
,
Raichurkar, Anandkumar
,
Kedari, Chaitanyakumar
,
Sharma, Sreevalli
,
Mudugal, Naina V
,
Narayan, Ashwini
,
Naveen Kumar, C. N
,
Nanduri, Robert
,
Bharath, Sowmya
,
Reddy, Jitendar
,
Panduga, Vijender
,
Prabhakar, K. R
,
Kandaswamy, Karthikeyan
,
Saralaya, Ramanatha
,
Kaur, Parvinder
,
Dinesh, Neela
,
Guptha, Supreeth
,
Rich, Kirsty
,
Murray, David
,
Plant, Helen
,
Preston, Marian
,
Ashton, Helen
,
Plant, Darren
,
Walsh, Jarrod
,
Alcock, Peter
,
Naylor, Kathryn
,
Collier, Matthew
,
Whiteaker, James
,
McLaughlin, Robert E
,
Mallya, Meenakshi
,
Panda, Manoranjan
,
Rudrapatna, Suresh
,
Ramachandran, Vasanthi
,
Shandil, Radha
,
Sambandamurthy, Vasan K
,
Mdluli, Khisi
,
Cooper, Christopher B
,
Rubin, Harvey
,
Yano, Takahiro
,
Iyer, Pravin
,
Narayanan, Shridhar
,
Kavanagh, Stefan
,
Mukherjee, Kakoli
,
Balasubramanian, V
,
Hosagrahara, Vinayak P
,
Solapure, Suresh
,
Ravishankar, Sudha
,
Hameed P, Shahul
Published in
Journal of medicinal chemistry
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4‑Aminoquinolone Piperidine Amides: Noncovalent Inhibitors of DprE1 with Long Residence Time and Potent Antimycobacterial Activity
by
Naik, Maruti
,
Humnabadkar, Vaishali
,
Tantry, Subramanyam J
,
Panda, Manoranjan
,
Narayan, Ashwini
,
Guptha, Supreeth
,
Panduga, Vijender
,
Manjrekar, Praveena
,
Jena, Lalit kumar
,
Koushik, Krishna
,
Shanbhag, Gajanan
,
Jatheendranath, Sandesh
,
Manjunatha, M. R
,
Gorai, Gopinath
,
Bathula, Chandramohan
,
Rudrapatna, Suresh
,
Achar, Vijayashree
,
Sharma, Sreevalli
,
Ambady, Anisha
,
Hegde, Naina
,
Mahadevaswamy, Jyothi
,
Kaur, Parvinder
,
Sambandamurthy, Vasan K
,
Awasthy, Disha
,
Narayan, Chandan
,
Ravishankar, Sudha
,
Madhavapeddi, Prashanti
,
Reddy, Jitendar
,
Prabhakar, KR
,
Saralaya, Ramanatha
,
Chatterji, Monalisa
,
Whiteaker, James
,
McLaughlin, Bob
,
Chiarelli, Laurent R
,
Riccardi, Giovanna
,
Pasca, Maria Rosalia
,
Binda, Claudia
,
Neres, João
,
Dhar, Neeraj
,
Signorino-Gelo, François
,
McKinney, John D
,
Ramachandran, Vasanthi
,
Shandil, Radha
,
Tommasi, Ruben
,
Iyer, Pravin S
,
Narayanan, Shridhar
,
Hosagrahara, Vinayak
,
Kavanagh, Stefan
,
Dinesh, Neela
,
Ghorpade, Sandeep R
Published in
Journal of medicinal chemistry
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6
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Discovery of benzothiazoles as antimycobacterial agents: Synthesis, structure–activity relationships and binding studies with Mycobacterium tuberculosis decaprenylphosphoryl-β-d-ri...
by
Landge, Sudhir
,
Mullick, Amrita B.
,
Nagalapur, Kavitha
,
Neres, João
,
Subbulakshmi, Venkita
,
Murugan, Kannan
,
Ghosh, Anirban
,
Sadler, Claire
,
Fellows, Mick D.
,
Humnabadkar, Vaishali
,
Mahadevaswamy, Jyothi
,
Vachaspati, Prakash
,
Sharma, Sreevalli
,
Kaur, Parvinder
,
Mallya, Meenakshi
,
Rudrapatna, Suresh
,
Awasthy, Disha
,
Sambandamurthy, Vasan K.
,
Pojer, Florence
,
Cole, Stewart T.
,
Balganesh, Tanjore S.
,
Ugarkar, Bheemarao G.
,
Balasubramanian, V.
,
Bandodkar, Balachandra S.
,
Panda, Manoranjan
,
Ramachandran, Vasanthi
Published in
Bioorganic & medicinal chemistry
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Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate
by
Hameed P, Shahul
,
Solapure, Suresh
,
Patil, Vikas
,
Henrich, Philipp P
,
Magistrado, Pamela A
,
Bharath, Sowmya
,
Murugan, Kannan
,
Viswanath, Pavithra
,
Puttur, Jayashree
,
Srivastava, Abhishek
,
Bellale, Eknath
,
Panduga, Vijender
,
Shanbag, Gajanan
,
Awasthy, Disha
,
Landge, Sudhir
,
Morayya, Sapna
,
Koushik, Krishna
,
Saralaya, Ramanatha
,
Raichurkar, Anandkumar
,
Rautela, Nikhil
,
Roy Choudhury, Nilanjana
,
Ambady, Anisha
,
Nandishaiah, Radha
,
Reddy, Jitendar
,
Prabhakar, K R
,
Menasinakai, Sreenivasaiah
,
Rudrapatna, Suresh
,
Chatterji, Monalisa
,
Jiménez-Díaz, María Belén
,
Martínez, María Santos
,
Sanz, Laura María
,
Coburn-Flynn, Olivia
,
Fidock, David A
,
Lukens, Amanda K
,
Wirth, Dyann F
,
Bandodkar, Balachandra
,
Mukherjee, Kakoli
,
McLaughlin, Robert E
,
Waterson, David
,
Rosenbrier-Ribeiro, Lyn
,
Hickling, Kevin
,
Balasubramanian, V
,
Warner, Peter
,
Hosagrahara, Vinayak
,
Dudley, Adam
,
Iyer, Pravin S
,
Narayanan, Shridhar
,
Kavanagh, Stefan
,
Sambandamurthy, Vasan K
Published in
Nature communications
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Thiazolopyridine Ureas as Novel Antitubercular Agents Acting through Inhibition of DNA Gyrase B
by
Kale, Manoj G
,
Raichurkar, Anandkumar
,
P, Shahul Hameed
,
Waterson, David
,
McKinney, David
,
Manjunatha, M. R
,
Kranthi, Usha
,
Koushik, Krishna
,
Jena, Lalit kumar
,
Shinde, Vikas
,
Rudrapatna, Suresh
,
Barde, Shubhada
,
Humnabadkar, Vaishali
,
Madhavapeddi, Prashanti
,
Basavarajappa, Halesha
,
Ghosh, Anirban
,
Ramya, VK
,
Guptha, Supreeth
,
Sharma, Sreevalli
,
Vachaspati, Prakash
,
Kumar, K.N. Mahesh
,
Giridhar, Jayashree
,
Reddy, Jitendar
,
Panduga, Vijender
,
Ganguly, Samit
,
Ahuja, Vijaykamal
,
Gaonkar, Sheshagiri
,
Kumar, C. N. Naveen
,
Ogg, Derek
,
Tucker, Julie A
,
Boriack-Sjodin, P. Ann
,
de Sousa, Sunita M
,
Sambandamurthy, Vasan K
,
Ghorpade, Sandeep R
Published in
Journal of medicinal chemistry
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Genetic and chemical validation identifies Mycobacterium tuberculosis topoisomerase I as an attractive anti-tubercular target
by
Ravishankar, Sudha
,
Ambady, Anisha
,
Awasthy, Disha
,
Mudugal, Naina Vinay
,
Menasinakai, Sreenivasaiah
,
Jatheendranath, Sandesh
,
Guptha, Supreeth
,
Sharma, Sreevalli
,
Balakrishnan, Gayathri
,
Nandishaiah, Radha
,
Ramachandran, Vasanthi
,
Eyermann, Charles J
,
Reck, Folkert
,
Rudrapatna, Suresh
,
Sambandamurthy, Vasan K
,
Sharma, Umender K
Published in
Tuberculosis (Edinburgh, Scotland)
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Scaffold morphing leading to evolution of 2,4-diaminoquinolines and aminopyrazolopyrimidines as inhibitors of the ATP synthesis pathway
by
Tantry, Subramanyam J.
,
Shinde, Vikas
,
Balakrishnan, Gayathri
,
Markad, Shankar D.
,
Gupta, Amit K.
,
Bhat, Jyothi
,
Narayan, Ashwini
,
Raichurkar, Anandkumar
,
Jena, Lalit Kumar
,
Sharma, Sreevalli
,
Kumar, Naveen
,
Nanduri, Robert
,
Bharath, Sowmya
,
Reddy, Jitendar
,
Panduga, Vijender
,
Prabhakar, K. R.
,
Kandaswamy, Karthikeyan
,
Kaur, Parvinder
,
Dinesh, Neela
,
Guptha, Supreeth
,
Saralaya, Ramanatha
,
Panda, Manoranjan
,
Rudrapatna, Suresh
,
Mallya, Meenakshi
,
Rubin, Harvey
,
Yano, Takahiro
,
Mdluili, Khisi
,
Cooper, Christopher B.
,
Balasubramanian, V.
,
Sambandamurthy, Vasan K.
,
Ramachandran, Vasanthi
,
Shandil, Radha
,
Kavanagh, Stefan
,
Narayanan, Shridhar
,
Iyer, Pravin
,
Mukherjee, Kakoli
,
Hosagrahara, Vinayak P.
,
Solapure, Suresh
,
Hameed P, Shahul
,
Ravishankar, Sudha
Published in
MedChemComm
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Scaffold morphing leading to evolution of 2,4-diaminoquinolines and aminopyrazolopyrimidines as inhibitors of the ATP synthesis pathwayThe authors declare no competing interests.El...
by
Tantry, Subramanyam J
,
Shinde, Vikas
,
Balakrishnan, Gayathri
,
Markad, Shankar D
,
Gupta, Amit K
,
Bhat, Jyothi
,
Narayan, Ashwini
,
Raichurkar, Anandkumar
,
Jena, Lalit Kumar
,
Sharma, Sreevalli
,
Kumar, Naveen
,
Nanduri, Robert
,
Bharath, Sowmya
,
Reddy, Jitendar
,
Panduga, Vijender
,
Prabhakar, K. R
,
Kandaswamy, Karthikeyan
,
Kaur, Parvinder
,
Dinesh, Neela
,
Guptha, Supreeth
,
Saralaya, Ramanatha
,
Panda, Manoranjan
,
Rudrapatna, Suresh
,
Mallya, Meenakshi
,
Rubin, Harvey
,
Yano, Takahiro
,
Mdluili, Khisi
,
Cooper, Christopher B
,
Balasubramanian, V
,
Sambandamurthy, Vasan K
,
Ramachandran, Vasanthi
,
Shandil, Radha
,
Kavanagh, Stefan
,
Narayanan, Shridhar
,
Iyer, Pravin
,
Mukherjee, Kakoli
,
Hosagrahara, Vinayak P
,
Solapure, Suresh
,
Hameed P, Shahul
,
Ravishankar, Sudha
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