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Search Results - Sivits, Jr, Glenn
Search Results - Sivits, Jr, Glenn
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Glucagon receptor antagonist-mediated improvements in glycemic control are dependent on functional pancreatic GLP-1 receptor
by
Gu, Wei
,
Winters, Katherine A
,
Motani, Alykhan S
,
Komorowski, Renée
,
Zhang, Ying
,
Liu, Qingxiang
,
Wu, Xiaosu
,
Rulifson, Ingrid C
,
Sivits, Jr, Glenn
,
Graham, Melissa
,
Yan, Hai
,
Wang, Paul
,
Moore, Steve
,
Meng, Tina
,
Lindberg, Richard A
,
Véniant, Murielle M
Published in
American journal of physiology: endocrinology and metabolism
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Pharmacological targeting of glucagon and glucagon-like peptide 1 receptors has different effects on energy state and glucose homeostasis in diet-induced obese mice
by
Gu, Wei
,
Lloyd, David J
,
Chinookswong, Narumol
,
Komorowski, Renée
,
Sivits, Jr, Glenn
,
Graham, Melissa
,
Winters, Katherine A
,
Yan, Hai
,
Boros, Laszlo G
,
Lindberg, Richard A
,
Véniant, Murielle M
Published in
The Journal of pharmacology and experimental therapeutics
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Antidiabetic effects of glucokinase regulatory protein small-molecule disruptors
by
Lloyd, David J
,
St Jean, Jr, David J
,
Kurzeja, Robert J M
,
Wahl, Robert C
,
Michelsen, Klaus
,
Cupples, Rod
,
Chen, Michelle
,
Wu, John
,
Sivits, Glenn
,
Helmering, Joan
,
Komorowski, Renée
,
Ashton, Kate S
,
Pennington, Lewis D
,
Fotsch, Christopher
,
Vazir, Mukta
,
Chen, Kui
,
Chmait, Samer
,
Zhang, Jiandong
,
Liu, Longbin
,
Norman, Mark H
,
Andrews, Kristin L
,
Bartberger, Michael D
,
Van, Gwyneth
,
Galbreath, Elizabeth J
,
Vonderfecht, Steven L
,
Wang, Minghan
,
Jordan, Steven R
,
Véniant, Murielle M
,
Hale, Clarence
Published in
Nature (London)
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Small Molecule Disruptors of the Glucokinase–Glucokinase Regulatory Protein Interaction: 1. Discovery of a Novel Tool Compound for in Vivo Proof-of-Concept
by
Ashton, Kate S.
,
Andrews, Kristin L.
,
Bryan, Marion C.
,
Chen, Jie
,
Chen, Kui
,
Chen, Michelle
,
Chmait, Samer
,
Croghan, Michael
,
Cupples, Rod
,
Fotsch, Christopher
,
Helmering, Joan
,
Jordan, Steve R.
,
Kurzeja, Robert J. M.
,
Michelsen, Klaus
,
Pennington, Lewis D.
,
Poon, Steve F.
,
Sivits, Glenn
,
Van, Gwyneth
,
Vonderfecht, Steve L.
,
Wahl, Robert C.
,
Zhang, Jiandong
,
Lloyd, David J.
,
Hale, Clarence
,
St. Jean, David J.
Published in
Journal of medicinal chemistry
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Small Molecule Disruptors of the Glucokinase–Glucokinase Regulatory Protein Interaction: 3. Structure–Activity Relationships within the Aryl Carbinol Region of the N‑Arylsulfonamid...
by
Nishimura, Nobuko
,
Norman, Mark H
,
Liu, Longbin
,
Yang, Kevin C
,
Ashton, Kate S
,
Bartberger, Michael D
,
Chmait, Samer
,
Chen, Jie
,
Cupples, Rod
,
Fotsch, Christopher
,
Helmering, Joan
,
Jordan, Steven R
,
Kunz, Roxanne K
,
Pennington, Lewis D
,
Poon, Steve F
,
Siegmund, Aaron
,
Sivits, Glenn
,
Lloyd, David J
,
Hale, Clarence
,
St. Jean, David J
Published in
Journal of medicinal chemistry
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Discovery and Structure-Guided Optimization of Diarylmethanesulfonamide Disrupters of Glucokinase–Glucokinase Regulatory Protein (GK–GKRP) Binding: Strategic Use of a N → S (nN → σ...
by
Pennington, Lewis D
,
Bartberger, Michael D
,
Croghan, Michael D
,
Andrews, Kristin L
,
Ashton, Kate S
,
Bourbeau, Matthew P
,
Chen, Jie
,
Chmait, Samer
,
Cupples, Rod
,
Fotsch, Christopher
,
Helmering, Joan
,
Hong, Fang-Tsao
,
Hungate, Randall W
,
Jordan, Steven R
,
Kong, Ke
,
Liu, Longbin
,
Michelsen, Klaus
,
Moyer, Carolyn
,
Nishimura, Nobuko
,
Norman, Mark H
,
Reichelt, Andreas
,
Siegmund, Aaron C
,
Sivits, Glenn
,
Tadesse, Seifu
,
Tegley, Christopher M
,
Van, Gwyneth
,
Yang, Kevin C
,
Yao, Guomin
,
Zhang, Jiandong
,
Lloyd, David J
,
Hale, Clarence
,
St. Jean, David J
Published in
Journal of medicinal chemistry
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Small Molecule Disruptors of the Glucokinase–Glucokinase Regulatory Protein Interaction: 5. A Novel Aryl Sulfone Series, Optimization Through Conformational Analysis
by
Tamayo, Nuria A
,
Norman, Mark H
,
Bartberger, Michael D
,
Hong, Fang-Tsao
,
Bo, Yunxin
,
Liu, Longbin
,
Nishimura, Nobuko
,
Yang, Kevin C
,
Tadesse, Seifu
,
Fotsch, Christopher
,
Chen, Jie
,
Chmait, Samer
,
Cupples, Rod
,
Hale, Clarence
,
Jordan, Steven R
,
Lloyd, David J
,
Sivits, Glenn
,
Van, Gwyneth
,
St. Jean, David J
Published in
Journal of medicinal chemistry
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Small Molecule Disruptors of the Glucokinase–Glucokinase Regulatory Protein Interaction: 2. Leveraging Structure-Based Drug Design to Identify Analogues with Improved Pharmacokinet...
by
St. Jean, David J.
,
Ashton, Kate S.
,
Bartberger, Michael D.
,
Chen, Jie
,
Chmait, Samer
,
Cupples, Rod
,
Galbreath, Elizabeth
,
Helmering, Joan
,
Hong, Fang-Tsao
,
Jordan, Steven R.
,
Liu, Longbin
,
Kunz, Roxanne K.
,
Michelsen, Klaus
,
Nishimura, Nobuko
,
Pennington, Lewis D.
,
Poon, Steve F.
,
Reid, Darren
,
Sivits, Glenn
,
Stec, Markian M.
,
Tadesse, Seifu
,
Tamayo, Nuria
,
Van, Gwyneth
,
Yang, Kevin C.
,
Zhang, Jiandong
,
Norman, Mark H.
,
Fotsch, Christopher
,
Lloyd, David J.
,
Hale, Clarence
Published in
Journal of medicinal chemistry
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Small Molecule Disruptors of the Glucokinase–Glucokinase Regulatory Protein Interaction: 4. Exploration of a Novel Binding Pocket
by
Hong, Fang-Tsao
,
Norman, Mark H
,
Ashton, Kate S
,
Bartberger, Michael D
,
Chen, Jie
,
Chmait, Samer
,
Cupples, Rod
,
Fotsch, Christopher
,
Jordan, Steven R
,
Lloyd, David J
,
Sivits, Glenn
,
Tadesse, Seifu
,
Hale, Clarence
,
St. Jean, David J
Published in
Journal of medicinal chemistry
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