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Synthesis, characterization, and first successful monkey imaging studies of metabotropic glutamate receptor subtype 5 (mGluR5) PET radiotracers
by
Hamill, Terence G.
,
Krause, Stephen
,
Ryan, Christine
,
Bonnefous, Celine
,
Govek, Steve
,
Seiders, T. Jon
,
Cosford, Nicholas D.P.
,
Roppe, Jeffrey
,
Kamenecka, Ted
,
Patel, Shil
,
Gibson, Raymond E.
,
Sanabria, Sandra
,
Riffel, Kerry
,
Eng, Waisi
,
King, Christopher
,
Yang, Xiaoqing
,
Green, Mitchell D.
,
O'malley, Stacey S.
,
Hargreaves, Richard
,
Burns, H. Donald
Published in
Synapse (New York, N.Y.)
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A novel, orally active LPA 1 receptor antagonist inhibits lung fibrosis in the mouse bleomycin model
by
Swaney, JS
,
Chapman, C
,
Correa, LD
,
Stebbins, KJ
,
Bundey, RA
,
Prodanovich, PC
,
Fagan, P
,
Baccei, CS
,
Santini, AM
,
Hutchinson, JH
,
Seiders, TJ
,
Parr, TA
,
Prasit, P
,
Evans, JF
,
Lorrain, DS
Published in
British journal of pharmacology
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Enantioselective Ruthenium-Catalyzed Ring-Closing Metathesis
by
Seiders, T. Jon
,
Ward, D. William
,
Grubbs, Robert H
Published in
Organic letters
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Structure/Energy Correlation of Bowl Depth and Inversion Barrier in Corannulene Derivatives: Combined Experimental and Quantum Mechanical Analysis
by
Seiders, T. Jon
,
Baldridge, Kim K
,
Grube, Gunther H
,
Siegel, Jay S
Published in
Journal of the American Chemical Society
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A novel, orally active LPA1 receptor antagonist inhibits lung fibrosis in the mouse bleomycin model
by
Swaney, JS
,
Chapman, C
,
Correa, LD
,
Stebbins, KJ
,
Bundey, RA
,
Prodanovich, PC
,
Fagan, P
,
Baccei, CS
,
Santini, AM
,
Hutchinson, JH
,
Seiders, TJ
,
Parr, TA
,
Prasit, P
,
Evans, JF
,
Lorrain, DS
Published in
British journal of pharmacology
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[ 3H]-Methoxymethyl-MTEP and [ 3H]-Methoxy-PEPy: potent and selective radioligands for the metabotropic glutamate subtype 5 (mGlu5) receptor
by
Cosford, Nicholas D.P
,
Roppe, Jeffrey
,
Tehrani, Lida
,
Schweiger, Edwin J
,
Seiders, T.Jon
,
Chaudary, Ashok
,
Rao, Sara
,
Varney, Mark A
Published in
Bioorganic & medicinal chemistry letters
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Synthesis of Corannulene and Alkyl Derivatives of Corannulene
by
Seiders, T. Jon
,
Elliott, Eric L
,
Grube, Gunther H
,
Siegel, Jay S
Published in
Journal of the American Chemical Society
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Synthesis and Quantum Mechanical Structure of sym-Pentamethylcorannulene and Decamethylcorannulene
by
Seiders, T. Jon
,
Baldridge, Kim K
,
Elliott, Eric L
,
Grube, Gunther H
,
Siegel, Jay S
Published in
Journal of the American Chemical Society
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Hexahapto Metal Coordination to Curved Polyaromatic Hydrocarbon Surfaces: The First Transition Metal Corannulene Complex
by
Seiders, T. Jon
,
Baldridge, Kim K
,
O'Connor, Joseph M
,
Siegel, Jay S
Published in
Journal of the American Chemical Society
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Synthesis and Characterization of the First Corannulene Cyclophane
by
Seiders, T. Jon
,
Baldridge, Kim K
,
Siegel, Jay S
Published in
Journal of the American Chemical Society
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Ionization of corannulene and 1,6-dimethylcorannulene: photoelectron spectra, electrochemistry, charge transfer bands and ab initio computations
by
Seiders, T.Jon
,
Baldridge, Kim K
,
Siegel, Jay S
,
Gleiter, Rolf
Published in
Tetrahedron letters
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3-[Substituted]-5-(5-pyridin-2-yl-2 H-tetrazol-2-yl)benzonitriles: Identification of highly potent and selective metabotropic glutamate subtype 5 receptor antagonists
by
Tehrani, Lida R.
,
Smith, Nicholas D.
,
Huang, Dehua
,
Poon, Steve F.
,
Roppe, Jeffrey R.
,
Seiders, Thomas Jon
,
Chapman, Deborah F.
,
Chung, Janice
,
Cramer, Merryl
,
Cosford, Nicholas D.P.
Published in
Bioorganic & medicinal chemistry letters
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