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Search Results - SUN, Shaiu-Ching
Search Results - SUN, Shaiu-Ching
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Pharmacological comparison of muscarinic ligands : Historical versus more recent muscarinic M1-preferring receptor agonists
by
HEINRICH, Julia N
,
BUTERA, John A
,
TSENG, Eugene
,
UVEGES, Albert J
,
MAYER, Scott C
,
CARRICK, Tikva
,
KRAMER, Angela
,
KOWAL, Dianne
,
LOCK, Tim
,
MARQUIS, Karen L
,
PAUSCH, Mark H
,
POPIOLEK, Mike
,
SUN, Shaiu-Ching
Published in
European journal of pharmacology
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Begacestat (GSI-953): a novel, selective thiophene sulfonamide inhibitor of amyloid precursor protein gamma-secretase for the treatment of Alzheimer's disease
by
Martone, Robert L
,
Zhou, Hua
,
Atchison, Kevin
,
Comery, Thomas
,
Xu, Jane Z
,
Huang, Xinyi
,
Gong, Xioahai
,
Jin, Mei
,
Kreft, Anthony
,
Harrison, Boyd
,
Mayer, Scott C
,
Aschmies, Suzan
,
Gonzales, Cathleen
,
Zaleska, Margaret M
,
Riddell, David R
,
Wagner, Erik
,
Lu, Peimin
,
Sun, Shaiu-Ching
,
Sonnenberg-Reines, June
,
Oganesian, Aram
,
Adkins, Karissa
,
Leach, Michael W
,
Clarke, David W
,
Huryn, Donna
,
Abou-Gharbia, Magid
,
Magolda, Ronald
,
Bard, Jonathan
,
Frick, Glen
,
Raje, Sangeeta
,
Forlow, S Bradley
,
Balliet, Carrie
,
Burczynski, Michael E
,
Reinhart, Peter H
,
Wan, Hong I
,
Pangalos, Menelas N
,
Jacobsen, J Steven
Published in
The Journal of pharmacology and experimental therapeutics
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Discovery of Begacestat, a Notch-1-Sparing γ-Secretase Inhibitor for the Treatment of Alzheimer’s Disease
by
Mayer, Scott C
,
Kreft, Anthony F
,
Harrison, Boyd
,
Abou-Gharbia, Magid
,
Antane, Madelene
,
Aschmies, Suzan
,
Atchison, Kevin
,
Chlenov, Michael
,
Cole, Derek C
,
Comery, Thomas
,
Diamantidis, George
,
Ellingboe, John
,
Fan, Kristi
,
Galante, Rocco
,
Gonzales, Cathleen
,
Ho, Douglas M
,
Hoke, Molly E
,
Hu, Yun
,
Huryn, Donna
,
Jain, Uday
,
Jin, Mei
,
Kremer, Kenneth
,
Kubrak, Dennis
,
Lin, Melissa
,
Lu, Peimin
,
Magolda, Ron
,
Martone, Robert
,
Moore, William
,
Oganesian, Aram
,
Pangalos, Menelas N
,
Porte, Alex
,
Reinhart, Peter
,
Resnick, Lynn
,
Riddell, David R
,
Sonnenberg-Reines, June
,
Stock, Joseph R
,
Sun, Shaiu-Ching
,
Wagner, Erik
,
Wang, Ting
,
Woller, Kevin
,
Xu, Zheng
,
Zaleska, Margaret M
,
Zeldis, Joseph
,
Zhang, Minsheng
,
Zhou, Hua
,
Jacobsen, J. Steven
Published in
Journal of medicinal chemistry
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Discovery of a novel series of Notch-sparing γ-secretase inhibitors
by
Kreft, Anthony
,
Harrison, Boyd
,
Aschmies, Suzan
,
Atchison, Kevin
,
Casebier, David
,
Cole, Derek C.
,
Diamantidis, George
,
Ellingboe, John
,
Hauze, Diane
,
Hu, Yun
,
Huryn, Donna
,
Jin, Mei
,
Kubrak, Dennis
,
Lu, Peimin
,
Lundquist, Joseph
,
Mann, Charles
,
Martone, Robert
,
Moore, William
,
Oganesian, Aram
,
Porte, Alex
,
Riddell, Dave R.
,
Sonnenberg-Reines, June
,
Stock, Joseph R.
,
Sun, Shaiu-Ching
,
Wagner, Erik
,
Woller, Kevin
,
Xu, Zheng
,
Zhou, Hua
,
Steven Jacobsen, J.
Published in
Bioorganic & medicinal chemistry
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( S) -N-(5-Chlorothiophene-2-sulfonyl)-β,β-diethylalaninol a Notch-1-sparing γ-secretase inhibitor
by
Cole, Derek C.
,
Stock, Joseph R.
,
Kreft, Anthony F.
,
Antane, Madelene
,
Aschmies, Suzan H.
,
Atchison, Kevin P.
,
Casebier, David S.
,
Comery, Thomas A.
,
Diamantidis, George
,
Ellingboe, John W.
,
Harrison, Boyd L.
,
Hu, Yun
,
Jin, Mei
,
Kubrak, Dennis M.
,
Lu, Peimin
,
Mann, Charles W.
,
Martone, Robert L.
,
Moore, William J.
,
Oganesian, Aram
,
Riddell, David R.
,
Sonnenberg-Reines, June
,
Sun, Shaiu-Ching
,
Wagner, Erik
,
Wang, Zheng
,
Woller, Kevin R.
,
Xu, Zheng
,
Zhou, Hua
,
Jacobsen, J. Steven
Published in
Bioorganic & medicinal chemistry letters
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Synthesis and structure–activity relationship of a novel series of heterocyclic sulfonamide γ-secretase inhibitors
by
Pu, Jun
,
Kreft, Anthony F.
,
Aschmies, Suzan H.
,
Atchison, Kevin P.
,
Berkowitz, Joshua
,
Caggiano, Thomas J.
,
Chlenov, Micheal
,
Diamantidis, George
,
Harrison, Boyd L.
,
Hu, Yun
,
Huryn, Donna
,
Steven Jacobsen, J.
,
Jin, Mei
,
Lipinski, Kerri
,
Lu, Peimin
,
Martone, Robert L.
,
Morris, Koi
,
Sonnenberg-Reines, June
,
Riddell, Dave R.
,
Sabalski, Joan
,
Sun, Shaiu-Ching
,
Wagner, Erik
,
Wang, Yiqun
,
Xu, Zheng
,
Zhou, Hua
,
Resnick, Lynn
Published in
Bioorganic & medicinal chemistry
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7
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Molecular-modeling based design, synthesis, and activity of substituted piperidines as γ-secretase inhibitors
by
Gundersen, Eric
,
Fan, Kristi
,
Haas, Kimberly
,
Huryn, Donna
,
Steven Jacobsen, J.
,
Kreft, Anthony
,
Martone, Robert
,
Mayer, Scott
,
Sonnenberg-Reines, June
,
Sun, Shaiu-Ching
,
Zhou, Hua
Published in
Bioorganic & medicinal chemistry letters
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8
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Pharmacological Characterization of the Muscarinic Agonist (3R,4R)-3-(3-Hexylsulfanyl-pyrazin-2-yloxy)-1-aza-bicyclo[2.2.1]heptane (WAY-132983) in in Vitro and in Vivo Models of Ch...
by
Sullivan, Nicole R
,
Leventhal, Liza
,
Harrison, James
,
Smith, Valerie A
,
Cummons, Terri A
,
Spangler, Taylor B
,
Sun, Shaiu-Ching
,
Lu, Peimin
,
Uveges, Albert J
,
Strassle, Brian W
,
Piesla, Michael J
,
Ramdass, Rana
,
Barry, Alena
,
Schantz, Jonathan
,
Adams, William
,
Whiteside, Garth T
,
Adedoyin, Adedayo
,
Jones, Philip G
Published in
The Journal of pharmacology and experimental therapeutics
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9
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Pharmacological comparison of muscarinic ligands: Historical versus more recent muscarinic M 1-preferring receptor agonists
by
Heinrich, Julia N.
,
Butera, John A.
,
Carrick, Tikva
,
Kramer, Angela
,
Kowal, Dianne
,
Lock, Tim
,
Marquis, Karen L.
,
Pausch, Mark H.
,
Popiolek, Mike
,
Sun, Shaiu-Ching
,
Tseng, Eugene
,
Uveges, Albert J.
,
Mayer, Scott C.
Published in
European journal of pharmacology
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Article
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10
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Begacestat (GSI-953): A Novel, Selective Thiophene Sulfonamide Inhibitor of Amyloid Precursor Protein γ-Secretase for the Treatment of Alzheimer's Disease
by
Robert L. Martone
,
Hua Zhou
,
Kevin Atchison
,
Thomas Comery
,
Jane Z. Xu
,
Xinyi Huang
,
Xioahai Gong
,
Mei Jin
,
Anthony Kreft
,
Boyd Harrison
,
Scott C. Mayer
,
Suzan Aschmies
,
Cathleen Gonzales
,
Margaret M. Zaleska
,
David R. Riddell
,
Erik Wagner
,
Peimin Lu
,
Shaiu-Ching Sun
,
June Sonnenberg-Reines
,
Aram Oganesian
,
Karissa Adkins
,
Michael W. Leach
,
David W. Clarke
,
Donna Huryn
,
Magid Abou-Gharbia
,
Ronald Magolda
,
Jonathan Bard
,
Glen Frick
,
Sangeeta Raje
,
S. Bradley Forlow
,
Carrie Balliet
,
Michael E. Burczynski
,
Peter H. Reinhart
,
Hong I. Wan
,
Menelas N. Pangalos
,
J. Steven Jacobsen
Published in
The Journal of pharmacology and experimental therapeutics
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11
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P4-244: Discovery of a novel series of notch-sparing γ-secretase inhibitors
by
Harrison, Boyd L.
,
Kreft, Anthony
,
Aschmies, Susan
,
Atchison, Kevin
,
Cole, Derek
,
Ellingboe, John
,
Hauze, Diane
,
Hu, Yun
,
Huryn, Donna
,
Jin, Mei
,
Kubrak, Dennis
,
Lu, Peimin
,
Mann, Charles
,
Martone, Robert
,
Moore, William
,
Porte, Alex
,
Riddell, David
,
Sonnenberg-Reines, June
,
Stock, Joseph
,
Sun, Shaiu-Ching
,
Wagner, Erik
,
Woller, Kevin
,
Xu, Zheng
,
Zhou, Hua
,
Jacobsen, Steven
Published in
Alzheimer's & dementia
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