Showing
1 - 11
results of
11
Skip to content
VuFind
Log in
Library Catalogue Plus
Library
Subject guides
Databases
Referencing
Catalogue
Articles Plus
Keyword
Title
Author
Subject
Find
Advanced Search
Search Results - Rigoreau, Laurent J.M
Search Results - Rigoreau, Laurent J.M
Showing
1 - 11
results of
11
Refine Results
Sort
Relevance
Date Descending
Author
Title
1
Loading…
Synthesis, crystal structure determination, and biological properties of the DNA-dependent protein kinase (DNA-PK) inhibitor 3-cyano-6-hydrazonomethyl-5-(4-pyridyl)pyrid-[1 H]-2-on...
by
Stockley, Martin
,
Clegg, William
,
Fontana, Gabriele
,
Golding, Bernard T
,
Martin, Niall
,
Rigoreau, Laurent J.M
,
Smith, Graeme C.M
,
Griffin, Roger J
Published in
Bioorganic & medicinal chemistry letters
Get full text
Items that this one cites
Items that cite this one
Article
Save to List
Saved in:
2
Loading…
2,6-Disubstituted pyran-4-one and thiopyran-4-one inhibitors of DNA-Dependent protein kinase (DNA-PK)
by
Hollick, Jonathan J.
,
Golding, Bernard T.
,
Hardcastle, Ian R.
,
Martin, Niall
,
Richardson, Caroline
,
Rigoreau, Laurent J.M.
,
Smith, Graeme C.M.
,
Griffin, Roger J.
Published in
Bioorganic & medicinal chemistry letters
Get full text
Items that this one cites
Items that cite this one
Article
Save to List
Saved in:
3
Loading…
Discovery, Characterization, and Structure-Based Optimization of Small-Molecule In Vitro and In Vivo Probes for Human DNA Polymerase Theta
by
Stockley, Martin L.
,
Ferdinand, Amanda
,
Benedetti, Giovanni
,
Blencowe, Peter
,
Boyd, Susan M.
,
Calder, Mat
,
Charles, Mark D.
,
Edwardes, Lucy V.
,
Ekwuru, Tennyson
,
Finch, Harry
,
Galbiati, Alessandro
,
Geo, Lerin
,
Grande, Diego
,
Grinkevich, Vera
,
Holliday, Nicholas D.
,
Krajewski, Wojciech W.
,
MacDonald, Ellen
,
Majithiya, Jayesh B.
,
McCarron, Hollie
,
McWhirter, Claire L.
,
Patel, Viral
,
Pedder, Chris
,
Rajendra, Eeson
,
Ranzani, Marco
,
Rigoreau, Laurent J. M.
,
Robinson, Helen M. R.
,
Schaedler, Theresia
,
Sirina, Julija
,
Smith, Graeme C. M.
,
Swarbrick, Martin E.
,
Turnbull, Andrew P.
,
Willis, Simon
,
Heald, Robert A.
Published in
Journal of medicinal chemistry
Get full text
Items that this one cites
Items that cite this one
Article
Save to List
Saved in:
4
Loading…
Structure-Based Design of Potent and Selective Inhibitors of the Metabolic Kinase PFKFB3
by
Boyd, Scott
,
Brookfield, Joanna L
,
Critchlow, Susan E
,
Cumming, Iain A
,
Curtis, Nicola J
,
Debreczeni, Judit
,
Degorce, Sébastien L
,
Donald, Craig
,
Evans, Nicola J
,
Groombridge, Sam
,
Hopcroft, Philip
,
Jones, Neil P
,
Kettle, Jason G
,
Lamont, Scott
,
Lewis, Hilary J
,
MacFaull, Philip
,
McLoughlin, Sheila B
,
Rigoreau, Laurent J. M
,
Smith, James M
,
St-Gallay, Steve
,
Stock, Julie K
,
Turnbull, Andrew P
,
Wheatley, Edward R
,
Winter, Jon
,
Wingfield, Jonathan
Published in
Journal of medicinal chemistry
Get full text
Items that this one cites
Items that cite this one
Article
Save to List
Saved in:
5
Loading…
Morpholylureas are a new class of potent and selective inhibitors of the type 5 17-β-hydroxysteroid dehydrogenase (AKR1C3)
by
Flanagan, Jack U.
,
Atwell, Graham J.
,
Heinrich, Daniel M.
,
Brooke, Darby G.
,
Silva, Shevan
,
Rigoreau, Laurent J.M.
,
Trivier, Elisabeth
,
Turnbull, Andrew P.
,
Raynham, Tony
,
Jamieson, Stephen M.F.
,
Denny, William A.
Published in
Bioorganic & medicinal chemistry
Get full text
Items that this one cites
Items that cite this one
Article
Save to List
Saved in:
6
Loading…
Identification of a novel orally bioavailable ERK5 inhibitor with selectivity over p38α and BRD4
by
Myers, Stephanie M.
,
Miller, Duncan C.
,
Molyneux, Lauren
,
Arasta, Mercedes
,
Bawn, Ruth H.
,
Blackburn, Timothy J.
,
Cook, Simon J.
,
Edwards, Noel
,
Endicott, Jane A.
,
Golding, Bernard T.
,
Griffin, Roger J.
,
Hammonds, Tim
,
Hardcastle, Ian R.
,
Harnor, Suzannah J.
,
Heptinstall, Amy B.
,
Lochhead, Pamela A.
,
Martin, Mathew P.
,
Martin, Nick C.
,
Newell, David R.
,
Owen, Paul J.
,
Pang, Leon C.
,
Reuillon, Tristan
,
Rigoreau, Laurent J.M.
,
Thomas, Huw D.
,
Tucker, Julie A.
,
Wang, Lan-Zhen
,
Wong, Ai-Ching
,
Noble, Martin E.M.
,
Wedge, Stephen R.
,
Cano, Celine
Published in
European journal of medicinal chemistry
Get full text
Items that this one cites
Items that cite this one
Article
Save to List
Saved in:
7
Loading…
Structure-Based Design of Potent and Selective 2-(Quinazolin-2-yl)phenol Inhibitors of Checkpoint Kinase 2
by
Caldwell, John J
,
Welsh, Emma J
,
Matijssen, Cornelis
,
Anderson, Victoria E
,
Antoni, Laurent
,
Boxall, Kathy
,
Urban, Frederique
,
Hayes, Angela
,
Raynaud, Florence I
,
Rigoreau, Laurent J. M
,
Raynham, Tony
,
Aherne, G. Wynne
,
Pearl, Laurence H
,
Oliver, Antony W
,
Garrett, Michelle D
,
Collins, Ian
Published in
Journal of medicinal chemistry
Get full text
Items that this one cites
Items that cite this one
Article
Save to List
Saved in:
8
Loading…
3‑(3,4-Dihydroisoquinolin-2(1H)‑ylsulfonyl)benzoic Acids: Highly Potent and Selective Inhibitors of the Type 5 17-β-Hydroxysteroid Dehydrogenase AKR1C3
by
Jamieson, Stephen M. F
,
Brooke, Darby G
,
Heinrich, Daniel
,
Atwell, Graham J
,
Silva, Shevan
,
Hamilton, Emma J
,
Turnbull, Andrew P
,
Rigoreau, Laurent J. M
,
Trivier, Elisabeth
,
Soudy, Christelle
,
Samlal, Sharon S
,
Owen, Paul J
,
Schroeder, Ewald
,
Raynham, Tony
,
Flanagan, Jack U
,
Denny, William A
Published in
Journal of medicinal chemistry
Get full text
Items that this one cites
Items that cite this one
Article
Save to List
Saved in:
9
Loading…
Synthesis and structure-activity relationships for 1-(4-(piperidin-1-ylsulfonyl)phenyl)pyrrolidin-2-ones as novel non-carboxylate inhibitors of the aldo-keto reductase enzyme AKR1C...
by
Heinrich, Daniel M
,
Flanagan, Jack U
,
Jamieson, Stephen M F
,
Silva, Shevan
,
Rigoreau, Laurent J M
,
Trivier, Elisabeth
,
Raynham, Tony
,
Turnbull, Andrew P
,
Denny, William A
Published in
European journal of medicinal chemistry
Get full text
Items that this one cites
Items that cite this one
Article
Save to List
Saved in:
10
Loading…
Pyranone, Thiopyranone, and Pyridone Inhibitors of Phosphatidylinositol 3-Kinase Related Kinases. Structure−Activity Relationships for DNA-Dependent Protein Kinase Inhibition, and...
by
Hollick, Jonathan J
,
Rigoreau, Laurent J. M
,
Cano-Soumillac, Celine
,
Cockcroft, Xiaoling
,
Curtin, Nicola J
,
Frigerio, Mark
,
Golding, Bernard T
,
Guiard, Sophie
,
Hardcastle, Ian R
,
Hickson, Ian
,
Hummersone, Marc G
,
Menear, Keith A
,
Martin, Niall M. B
,
Matthews, Ian
,
Newell, David R
,
Ord, Rachel
,
Richardson, Caroline J
,
Smith, Graeme C. M
,
Griffin, Roger J
Published in
Journal of medicinal chemistry
Get full text
Items that this one cites
Items that cite this one
Article
Save to List
Saved in:
11
Loading…
Reactivity and Mechanism in the Hydrolysis of β-Sultams
by
Baxter, Nicholas J
,
Rigoreau, Laurent J. M
,
Laws, Andrew P
,
Page, Michael I
Published in
Journal of the American Chemical Society
Get full text
Items that this one cites
Items that cite this one
Article
Save to List
Saved in:
Search Tools:
RSS Feed
Email Search
Save Search
Back
Refine Results
Page will reload when a filter is selected or excluded.
Limit To
Peer Reviewed
11 results
11
Full Text
11 results
11
Format
Articles
11 results
11
Journal Title
Journal Of Medicinal Chemistry
5 results
5
Bioorganic & Medicinal Chemistry Letters
2 results
2
European Journal Of Medicinal Chemistry
2 results
2
Bioorganic & Medicinal Chemistry
1 results
1
Journal Of The American Chemical Society
1 results
1
Subjects
Science & Technology
11 results
11
Chemistry, Medicinal
10 results
10
Life Sciences & Biomedicine
10 results
10
Pharmacology & Pharmacy
10 results
10
Humans
8 results
8
Structure-Activity Relationship
8 results
8
Models, Molecular
6 results
6
Enzyme Inhibitors - Pharmacology
5 results
5
Animals
4 results
4
Chemistry
4 results
4
Enzyme Inhibitors - Chemistry
4 results
4
Physical Sciences
4 results
4
Protein-Serine-Threonine Kinases - Antagonists & Inhibitors
4 results
4
3-Hydroxysteroid Dehydrogenases - Antagonists & Inhibitors
3 results
3
Aldo-Keto Reductase Family 1 Member C3
3 results
3
Antineoplastic Agents - Pharmacology
3 results
3
Chemistry, Organic
3 results
3
Crystallography, X-Ray
3 results
3
Enzyme Inhibitors - Chemical Synthesis
3 results
3
Hydroxyprostaglandin Dehydrogenases - Antagonists & Inhibitors
3 results
3
Year of Publication
From:
To:
Source
Science Citation Index Expanded (Web Of Science)
11 results
11
Acs Crkn Legacy Archives
6 results
6
American Chemical Society:jisc Collections:american Chemical Society Read & Publish Agreement 2022-2024 (Reading List)
6 results
6
Elsevier Sciencedirect Journals
5 results
5
Sciencedirect Freedom Collection
5 results
5
Backfile Package - Organic Chemistry (Legacy) [Yco]
5 results
5