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Search Results - Ratia, Kiira M.
Search Results - Ratia, Kiira M.
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Isoquinoline Kelch-like ECH-Associated Protein 1‑Nuclear Factor (Erythroid-Derived 2)-like 2 (KEAP1-NRF2) Inhibitors with High Metabolic Stability
by
Lazzara, Phillip R
,
David, Brian P
,
Ankireddy, Aparna
,
Richardson, Benjamin G
,
Dye, Katherine
,
Ratia, Kiira M
,
Reddy, Sekhar P
,
Moore, Terry W
Published in
Journal of medicinal chemistry
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Mechanism of Allosteric Modulation of Nicotinamide Phosphoribosyltransferase to Elevate Cellular NAD
by
Ratia, Kiira M.
,
Shen, Zhengnan
,
Gordon-Blake, Jesse
,
Lee, Hyun
,
Laham, Megan S.
,
Krider, Isabella S.
,
Christie, Nicholas
,
Ackerman-Berrier, Martha
,
Penton, Christopher
,
Knowles, Natalie G.
,
Musku, Soumya Reddy
,
Fu, Jiqiang
,
Velma, Ganga Reddy
,
Xiong, Rui
,
Thatcher, Gregory R. J.
Published in
Biochemistry (Easton)
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Synthesis and Evaluation of Noncovalent Naphthalene-Based KEAP1-NRF2 Inhibitors
by
Lazzara, Phillip R
,
Jain, Atul D
,
Maldonado, Amanda C
,
Richardson, Benjamin
,
Skowron, Kornelia J
,
David, Brian P
,
Siddiqui, Zamia
,
Ratia, Kiira M
,
Moore, Terry W
Published in
ACS medicinal chemistry letters
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Discovery of Nonlipogenic ABCA1 Inducing Compounds with Potential in Alzheimer’s Disease and Type 2 Diabetes
by
Ben Aissa, Manel
,
Lewandowski, Cutler T
,
Ratia, Kiira M
,
Lee, Sue H
,
Layden, Brian T
,
LaDu, Mary Jo
,
Thatcher, Gregory R. J
Published in
ACS pharmacology & translational science
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Structural Basis for the Ubiquitin-Linkage Specificity and deISGylating activity of SARS-CoV papain-like protease
by
Ratia, Kiira
,
Kilianski, Andrew
,
Baez-Santos, Yahira M
,
Baker, Susan C
,
Mesecar, Andrew
Published in
PLoS pathogens
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PHY34 inhibits autophagy through V-ATPase V0A2 subunit inhibition and CAS/CSE1L nuclear cargo trafficking in high grade serous ovarian cancer
by
Salvi, Amrita
,
Young, Alexandria N
,
Huntsman, Andrew C
,
Pergande, Melissa R
,
Korkmaz, Melissa A
,
Rathnayake, Rathnayake A
,
Mize, Brittney K
,
Kinghorn, A Douglas
,
Zhang, Xiaoli
,
Ratia, Kiira
,
Schirle, Markus
,
Thomas, Jason R
,
Brittain, Scott M
,
Shelton, Claude
,
Aldrich, Leslie N
,
Cologna, Stephanie M
,
Fuchs, James R
,
Burdette, Joanna E
Published in
Cell death & disease
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Deubiquitinating and Interferon Antagonism Activities of Coronavirus Papain-Like Proteases
by
Clementz, Mark A
,
Chen, Zhongbin
,
Banach, Bridget S
,
Wang, Yanhua
,
Sun, Li
,
Ratia, Kiira
,
Baez-Santos, Yahira M
,
Wang, Jie
,
Takayama, Jun
,
Ghosh, Arun K
,
Li, Kui
,
Mesecar, Andrew D
,
Baker, Susan C
Published in
Journal of Virology
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Synthesis, Optimization, and Structure–Activity Relationships of Nicotinamide Phosphoribosyltransferase (NAMPT) Positive Allosteric Modulators (N-PAMs)
by
Shen, Zhengnan
,
Ratia, Kiira
,
Krider, Isabella
,
Ackerman-Berrier, Martha
,
Penton, Christopher
,
Musku, Soumya Reddy
,
Gordon-Blake, Jesse M.
,
Laham, Megan S.
,
Christie, Nicholas
,
Ma, Nina
,
Fu, Jiqiang
,
Xiong, Rui
,
Courey, Jenna M.
,
Velma, Ganga Reddy
,
Thatcher, Gregory R. J.
Published in
Journal of medicinal chemistry
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Novel Pyrrolopyridone Bromodomain and Extra-Terminal Motif (BET) Inhibitors Effective in Endocrine-Resistant ER+ Breast Cancer with Acquired Resistance to Fulvestrant and Palbocicl...
by
Li, Yangfeng
,
Zhao, Jiong
,
Gutgesell, Lauren M
,
Shen, Zhengnan
,
Ratia, Kiira
,
Dye, Katherine
,
Dubrovskyi, Oleksii
,
Zhao, Huiping
,
Huang, Fei
,
Tonetti, Debra A
,
Thatcher, Gregory R. J
,
Xiong, Rui
Published in
Journal of medicinal chemistry
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Design and Synthesis of Peptidomimetic Severe Acute Respiratory Syndrome Chymotrypsin-like Protease Inhibitors
by
Ghosh, Arun K
,
Xi, Kai
,
Ratia, Kiira
,
Santarsiero, Bernard D
,
Fu, Wentao
,
Harcourt, Brian H
,
Rota, Paul A
,
Baker, Susan C
,
Johnson, Michael E
,
Mesecar, Andrew D
Published in
Journal of medicinal chemistry
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Nicotinamide Phosphoribosyltransferase Positive Allosteric Modulators Attenuate Neuronal Oxidative Stress
by
Gordon-Blake, Jesse
,
Ratia, Kiira
,
Weidig, Victoria
,
Velma, Ganga Reddy
,
Ackerman-Berrier, Martha
,
Penton, Christopher
,
Musku, Soumya Reddy
,
Alves, Erick T.M.
,
Driver, Tom
,
Tai, Leon
,
Thatcher, Gregory R. J.
Published in
ACS medicinal chemistry letters
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Abstract 3910: Identification of lead organic compounds active against stem cell-like neuroblastoma cells by high throughput screening
by
Ikegaki, Naohiko
,
Ratia, Kiira
,
Hsiao, Ruth
,
Limpar, Mariko M.
,
Lomahan, Sarah
,
Tang, Xao X.
Published in
Cancer research (Chicago, Ill.)
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Structural Basis for the Ubiquitin-Linkage Specificity and deISGylating Activity of SARS-CoV Papain-Like Protease: e1004113
by
Ratia, Kiira
,
Kilianski, Andrew
,
Baez-Santos, Yahira M
,
Baker, Susan C
,
Mesecar, Andrew
Published in
PLoS pathogens
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Dual Inhibition of Cathepsin L and 3CL-Pro by GC-376 Constrains SARS Cov2 Infection Including Omicron Variant
by
Prabhakar, Bellur S
,
Prabhakaran Kumar
,
Ratia, Kiira
,
Richner, Justin M
,
Thatcher, Gregory R J
,
Kadam, Rashmi
,
Smieszek, Sandra P
,
Przychodzen, Bartlomiej P
,
Koprivica, Vuk
,
Birznieks, Gunther
,
Polymeropoulos, Mihael H
Published in
bioRxiv
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