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Search Results - RAMI, Harshad K
Search Results - RAMI, Harshad K
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Characterization of SB-705498, a Potent and Selective Vanilloid Receptor-1 (VR1/TRPV1) Antagonist That Inhibits the Capsaicin-, Acid-, and Heat-Mediated Activation of the Receptor
by
Gunthorpe, Martin J
,
Hannan, Sara Luis
,
Smart, Darren
,
Jerman, Jeffrey C
,
Arpino, Sandra
,
Smith, Graham D
,
Brough, Stephen
,
Wright, Jim
,
Egerton, Julie
,
Lappin, Sarah C
,
Holland, Vicky A
,
Winborn, Kim
,
Thompson, Mervyn
,
Rami, Harshad K
,
Randall, Andrew
,
Davis, John B
Published in
The Journal of pharmacology and experimental therapeutics
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Discovery of small molecule antagonists of TRPV1
by
RAMI, Harshad K
,
THOMPSON, Mervyn
,
DAVIS, John B
,
WYMAN, Paul
,
JERMAN, Jeffrey C
,
EGERTON, Julie
,
BROUGH, Stephen
,
STEVENS, Alexander J
,
RANDALL, Andrew D
,
SMART, Darren
,
GUNTHORPE, Martin J
Published in
Bioorganic & medicinal chemistry letters
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Discovery of SB-705498: A potent, selective and orally bioavailable TRPV1 antagonist suitable for clinical development
by
Rami, Harshad K.
,
Thompson, Mervyn
,
Stemp, Geoffrey
,
Fell, Steve
,
Jerman, Jeffrey C.
,
Stevens, Alexander J.
,
Smart, Darren
,
Sargent, Becky
,
Sanderson, Dominic
,
Randall, Andrew D.
,
Gunthorpe, Martin J.
,
Davis, John B.
Published in
Bioorganic & medicinal chemistry letters
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Design and synthesis of 6-phenylnicotinamide derivatives as antagonists of TRPV1
by
Westaway, Susan M.
,
Thompson, Mervyn
,
Rami, Harshad K.
,
Stemp, Geoffrey
,
Trouw, Leontine S.
,
Mitchell, Darren J.
,
Seal, Jon T.
,
Medhurst, Stephen J.
,
Lappin, Sarah C.
,
Biggs, James
,
Wright, James
,
Arpino, Sandra
,
Jerman, Jeffrey C.
,
Cryan, Jennifer E.
,
Holland, Vicky
,
Winborn, Kim Y.
,
Coleman, Tanya
,
Stevens, Alexander J.
,
Davis, John B.
,
Gunthorpe, Martin J.
Published in
Bioorganic & medicinal chemistry
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3,4-Dihydro-2H-benzoxazinones are 5-HT1A receptor antagonists with potent 5-HT reuptake inhibitory activity
by
ATKINSON, Peter J
,
BROMIDGE, Steven M
,
RAMI, Harshad K
,
RILEY, Graham J
,
SCOTT, Claire M
,
SHAW, Tracey E
,
STARR, Kathryn R
,
STEMP, Geoffrey
,
THEWLIS, Kevin M
,
THOMAS, David R
,
THOMPSON, Mervyn
,
VONG, Antonio K. K
,
DUXON, Mark S
,
WATSON, Jeannette M
,
GASTER, Laramie M
,
HADLEY, Michael S
,
HAMMOND, Beverley
,
JOHNSON, Christopher N
,
MIDDLEMISS, Derek N
,
NORTH, Stephanie E
,
PRICE, Gary W
Published in
Bioorganic & medicinal chemistry letters
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Non-thiazolidinedione antihyperglycaemic agents. Part 4: Synthesis of (±)-, ( R)-(+)- and ( S)-(−)-enantiomers of 2-oxy-3-arylpropanoic acids
by
Haigh, David
,
Birrell, Helen C
,
Cantello, Barrie C.C
,
Hindley, Richard M
,
Ramaswamy, Anantha
,
Rami, Harshad K
,
Stevens, Nicola C
Published in
Tetrahedron: asymmetry
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N-Tetrahydroquinolinyl, N-quinolinyl and N-isoquinolinyl biaryl carboxamides as antagonists of TRPV1
by
Westaway, Susan M.
,
Chung, Ying-Kit
,
Davis, John B.
,
Holland, Vicky
,
Jerman, Jeffrey C.
,
Medhurst, Stephen J.
,
Rami, Harshad K.
,
Stemp, Geoffrey
,
Stevens, Alexander J.
,
Thompson, Mervyn
,
Winborn, Kim Y.
,
Wright, James
Published in
Bioorganic & medicinal chemistry letters
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Evidence for a molecular mechanism of teratogenicity of SB-236057, a 5-HT1B receptor inverse agonist that alters axial formation
by
Augustine-Rauch, Karen A.
,
Zhang, Qin J.
,
Leonard, Jennifer L.
,
Chadderton, Antony
,
Welsh, Michael J.
,
Rami, Harshad K.
,
Thompson, Mervyn
,
Gaster, Laramie
,
Wier, Patrick J.
Published in
Birth defects research. A Clinical and molecular teratology
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Bioreductive fluorescent markers for hypoxic cells: a study of 2-nitroimidazoles with 1-substituents containing fluorescent, bridgehead-nitrogen, bicyclic systems
by
Hodgkiss, Richard J
,
Middleton, Richard W
,
Parrick, John
,
Rami, Harshad K
,
Wardman, Peter
,
Wilson, George D
Published in
Journal of medicinal chemistry
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The therapeutic potential of TRPV1 (VR1) antagonists: clinical answers await
by
Rami, Harshad K.
,
Gunthorpe, Martin J.
Published in
Drug discovery today. Therapeutic strategies
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11
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3,4-Dihydro-2H-benzoxazinones are 5-HT(1A) receptor antagonists with potent 5-HT reuptake inhibitory activity
by
Atkinson, Peter J
,
Bromidge, Steven M
,
Duxon, Mark S
,
Gaster, Laramie M
,
Hadley, Michael S
,
Hammond, Beverley
,
Johnson, Christopher N
,
Middlemiss, Derek N
,
North, Stephanie E
,
Price, Gary W
,
Rami, Harshad K
,
Riley, Graham J
,
Scott, Claire M
,
Shaw, Tracey E
,
Starr, Kathryn R
,
Stemp, Geoffrey
,
Thewlis, Kevin M
,
Thomas, David R
,
Thompson, Mervyn
,
Vong, Antonio K K
,
Watson, Jeannette M
Published in
Bioorganic & medicinal chemistry letters
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Non-thiazolidinedione antihyperglycaemic agents. Part 3: the effects of stereochemistry on the potency of α-methoxy-β-phenylpropanoic acids
by
Haigh, David
,
Allen, Graham
,
Birrell, Helen C.
,
Buckle, Derek R.
,
Cantello, Barrie C.C.
,
Eggleston, Drake S.
,
Haltiwanger, R.Curtis
,
Holder, Julie C.
,
Lister, Carolyn A.
,
Pinto, Ivan L.
,
Rami, Harshad K.
,
Sime, John T.
,
Smith, Stephen A.
,
Sweeney, John D.
Published in
Bioorganic & medicinal chemistry
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3,4-Dihydro-2 H-benzoxazinones are 5-HT 1A receptor antagonists with potent 5-HT reuptake inhibitory activity
by
Atkinson, Peter J.
,
Bromidge, Steven M.
,
Duxon, Mark S.
,
Gaster, Laramie M.
,
Hadley, Michael S.
,
Hammond, Beverley
,
Johnson, Christopher N.
,
Middlemiss, Derek N.
,
North, Stephanie E.
,
Price, Gary W.
,
Rami, Harshad K.
,
Riley, Graham J.
,
Scott, Claire M.
,
Shaw, Tracey E.
,
Starr, Kathryn R.
,
Stemp, Geoffrey
,
Thewlis, Kevin M.
,
Thomas, David R.
,
Thompson, Mervyn
,
Vong, Antonio K.K.
,
Watson, Jeannette M.
Published in
Bioorganic & medicinal chemistry letters
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14
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A hetero Diels-Alder approach to novel thiopyran analogues of aprikalim, A potassium channel activator
by
Pinto, Ivan L.
,
Buckle, Derek R.
,
Rami, Harshad K.
,
Smith, David G.
Published in
Tetrahedron letters
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15
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The Contribution of Classical (β1/2-) and Atypical β-Adrenoceptors to the Stimulation of Human White Adipocyte Lipolysis and Right Atrial Appendage Contraction by Novel β3-Adren...
by
Matthew V. Sennitt
,
Alberto J. Kaumann
,
Peter Molenaar
,
Lee J. Beeley
,
Paul W. Young
,
John Kelly
,
Helen Chapman
,
Sian M. Henson
,
John M. Berge
,
David K. Dean
,
Nikesh R. Kotecha
,
Helen K. A. Morgan
,
Harshad K. Rami
,
Robert W. Ward
,
Mervyn Thompson
,
Shelagh Wilson
,
Stephen A. Smith
,
Michael A. Cawthorne
,
Michael J. Stock
,
Jonathan R. S. Arch
Published in
The Journal of pharmacology and experimental therapeutics
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