MK-4815, a Potential New Oral Agent for Treatment of Malaria by POWLES, Mary Ann, ALLOCCO, John, YEUNG, Lai, NARE, Bakela, LIBERATOR, Paul, SCHMATZ, Dennis

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Broadening the Spectrum of β-Lactam Antibiotics through Inhibition of Signal Peptidase Type I by THERIEN, Alex G, HUBER, Joann L, XIN GU, KEVIN, Nancy J, LAFLEUR, Josiane, LEAVITT, Penny S, LEBEAU-JACOB, Christian, LEE, Suzy S, LIN, Molly M, MICHELS, Anna A, OGAWA, Aimie M, PAINTER, Ronald E, WILSON, Kenneth E, PARISH, Craig A, PARK, Young-Whan, BENTON-PERDOMO, Liliana, PETCU, Mihai, PHILLIPS, John W, POWLES, Mary Ann, SKOREY, Kathryn I, TAM, John, TAN, Christopher M, YOUNG, Katherine, BEAULIEU, Patrick, WONG, Simon, WADDELL, Sherman T, MIESEL, Lynn, CARON, Alexandre, CLAVEAU, David, DESCHAMPS, Kathleen, DONALD, Robert G. K, GALGOCI, Andrew M, GALLANT, Michel

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Design, Synthesis, and Evaluation of Novel and Selective G‑protein Coupled Receptor 120 (GPR120) Spirocyclic Agonists by Cox, Jason M, Chu, Hong D, Chelliah, Mariappan V, Debenham, John S, Eagen, Keith, Lan, Ping, Lombardo, Matthew, London, Clare, Plotkin, Michael A, Shah, Unmesh, Sun, Zhongxiang, Vaccaro, Henry M, Venkatraman, Srikanth, Suzuki, Takao, Wang, Nengxue, Ashley, Eric R, Crespo, Alejandro, Madeira, Maria, Leung, Dennis H, Alleyne, Candice, Ogawa, Aimie M, Souza, Sarah, Thomas-Fowlkes, Brande, Di Salvo, Jerry, Weinglass, Adam, Kirkland, Melissa, Pachanski, Michele, Powles, Mary Ann, Tozzo, Effie, Akiyama, Taro E, Ujjainwalla, Feroze, Tata, James R, Sinz, Christopher J

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Characterization of Plasmodium falciparum cGMP-dependent protein kinase ( PfPKG): Antiparasitic activity of a PKG inhibitor by Diaz, Carmen A., Allocco, John, Powles, Mary Ann, Yeung, Lai, Donald, Robert G.K., Anderson, Jennifer W., Liberator, Paul A.

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Efficacy of Caspofungin in a Juvenile Mouse Model of Central Nervous System Candidiasis by FLATTERY, Amy M, HICKEY, Emily, ABRUZZO, George K, GILL, Charles J, POWLES, Mary Ann, MISURA, Andrew S, GALGOCI, Andrew M, ELLIS, Joan D, RENA ZHANG, SANDHU, Punam, RONAN, John

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In Vivo Efficacy of Relebactam (MK-7655) in Combination with Imipenem-Cilastatin in Murine Infection Models by Powles, Mary Ann, Galgoci, Andrew, Misura, Andrew, Colwell, Lawrence, Dingley, Karen H, Tang, Wei, Wu, Jin, Blizzard, Timothy, Motyl, Mary, Young, Katherine

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MOLECULAR PHYLOGENY OF THE OTHER TISSUE COCCIDIA: LANKESTERELLA AND CARYOSPORA by Barta, JohnR, Martin, Donald S, Carreno, Ramon A, Siddall, Mark E, Profous-Juchelka, Helen, Hozza, Mark, Ann Powles, Mary, Sundermann, Christine

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Discovery of benzofuran propanoic acid GPR120 agonists: From uHTS hit to mechanism-based pharmacodynamic effects by Lombardo, Matthew, Bender, Kate, London, Clare, Plotkin, Michael A., Kirkland, Melissa, Mane, Joel, Pachanski, Michele, Geissler, Wayne, Cummings, John, Habulihaz, Bahanu, Akiyama, Taro E., Di Salvo, Jerry, Madeira, Maria, Pols, Joanna, Powles, Mary Ann, Finley, Michael F., Johnson, Eric, Roussel, Thomas, Uebele, Victor N., Crespo, Alejandro, Leung, Dennis, Alleyne, Candice, Trusca, Dorina, Lei, Ying, Howard, Andrew D., Ujjainwalla, Feroze, Tata, James R., Sinz, Christopher J.

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Discovery of Novel Tricyclic Heterocycles as Potent and Selective DPP‑4 Inhibitors for the Treatment of Type 2 Diabetes by Wu, Wen-Lian, Hao, Jinsong, Domalski, Martin, Burnett, Duane A, Pissarnitski, Dmitri, Zhao, Zhiqiang, Stamford, Andrew, Scapin, Giovanna, Gao, Ying-Duo, Soriano, Aileen, Kelly, Terri M, Yao, Zuliang, Powles, Mary Ann, Chen, Shiying, Mei, Hong, Hwa, Joyce

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Scaffold-hopping from xanthines to tricyclic guanines: A case study of dipeptidyl peptidase 4 (DPP4) inhibitors by Pissarnitski, Dmitri A., Zhao, Zhiqiang, Cole, David, Wu, Wen-Lian, Domalski, Martin, Clader, John W., Scapin, Giovanna, Voigt, Johannes, Soriano, Aileen, Kelly, Theresa, Powles, Mary Ann, Yao, Zuliang, Burnett, Duane A.

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Isolation and Structure Elucidation of Parnafungins, Antifungal Natural Products that Inhibit mRNA Polyadenylation by Parish, Craig A, Smith, Scott K, Calati, Kathleen, Zink, Deborah, Wilson, Kenneth, Roemer, Terry, Jiang, Bo, Xu, Deming, Bills, Gerald, Platas, Gonzalo, Peláez, Fernando, Díez, Maria Teresa, Tsou, Nancy, McKeown, Arlene E, Ball, Richard G, Powles, Mary Ann, Yeung, Lai, Liberator, Paul, Harris, Guy

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Corrigendum to “Discovery of benzofuran propanoic acid GPR120 agonists: From uHTS hit to mechanism-based pharmacodynamic effects” [Bioorg. Med. Chem. Lett. 26 (2016) 5724–5728]... by Lombardo, Matthew, Bender, Kate, London, Clare, Plotkin, Michael A., Kirkland, Melissa, Mane, Joel, Pachanski, Michele, Geissler, Wayne, Cummings, John, Habulihaz, Bahanu, Akiyama, Taro E., Di Salvo, Jerry, Madeira, Maria, Pols, Joanna, Powles, Mary Ann, Finley, Michael F., Johnson, Eric, Roussel, Thomas, Uebele, Victor N., Crespo, Alejandro, Leung, Dennis, Alleyne, Candice, Trusca, Dorina, Lei, Ying, Howard, Andrew D., Ujjainwalla, Feroze, Tata, James R., Sinz, Christopher J.

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Discovery and Optimization of a Novel Triazole Series of GPR142 Agonists for the Treatment of Type 2 Diabetes by Guo, Liangqin, Parker, Dann L, Zang, Yi, Sweis, Ramzi F, Liu, Weiguo, Sherer, Edward C, Buist, Nicole, Terebetski, Jenna, Kelly, Terri, Bugianesi, Randal, Priest, Birgit T, Dingley, Karen H, Li, Xiaofang, Mitelman, Stan, Salituro, Gino, Trujillo, Maria E, Pachanski, Michele, Kirkland, Melissa, Powles, Mary Ann, Eiermann, George J, Feng, Yue, Shang, Jin, Howard, Andrew D, Ujjainwalla, Feroze, Sinz, Christopher J, Debenham, John S, Edmondson, Scott D, Nargund, Ravi P, Hagmann, William K, Li, Derun

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Efficacy of MK-991 (L-743,872), a semisynthetic pneumocandin, in murine models of Pneumocystis carinii by POWLES, M. A, LIBERATOR, P, SCHMATZ, D, ANDERSON, J, KARKHANIS, Y, DROPINSKI, J. F, BOUFFARD, F. A, BALKOVEC, J. M, FUJIOKA, H, AIKAWA, M, MCFADDEN, D

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Efficacy of MK-991 (L-743,872), a Semisynthetic Pneumocandin, in Murine Models ofPneumocystis carinii by Powles, Mary Ann, Liberator, Paul, Anderson, Jennifer, Karkhanis, Yashwant, Dropinski, James F, Bouffard, F. Aileen, Balkovec, James M, Fujioka, Hisashi, Aikawa, Masamichi, McFadden, Diane, Schmatz, Dennis

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Potent 4-aminopiperidine based antimalarial agents by Brinner, Kristin M., Powles, Mary Ann, Schmatz, Dennis M., Ellman, Jonathan A.

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Corrigendum to “Potent 4-aminopiperidine based antimalarial agents” [Bioorg. Med. Chem. Lett. 15 (2005) 345] by Brinner, Kristin M., Powles, Mary Ann, Schmatz, Dennis M., Ellman, Jonathan A.

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Molecular Phylogeny of the Other Tissue Coccidia: Lankesterella and Caryospora by Barta, John. R., Martin, Donald S., Carreno, Ramon A., Siddall, Mark E., Profous-Juchelka, Helen, Hozza, Mark, Powles, Mary Ann, Sundermann, Christine

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Synthesis, stability, and biological evaluation of water-soluble prodrugs of a new echinocandin lipopeptide. Discovery of a potential clinical agent for the treatment of systemic c... by Balkovec, James M, Black, Regina M, Hammond, Milton L, Heck, James V, Zambias, Robert A, Abruzzo, George, Bartizal, Ken, Kropp, Helmut, Trainor, Charlotte

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An observational study showed that explaining randomization using gambling-related metaphors and computer-agency descriptions impeded randomized clinical trial recruitment by Jepson, Marcus, Elliott, Daisy, Conefrey, Carmel, Wade, Julia, Rooshenas, Leila, Wilson, Caroline, Beard, David, Blazeby, Jane M., Birtle, Alison, Halliday, Alison, Stein, Rob, Donovan, Jenny L., Beard, David, Carr, Andrew, Cook, Jonathan, Cooper, Cushla, Dean, Benjamin, Donovan, Jenny L., Gray, Alastair, Judge, Andrew, Merritt, Naomi, Moser, Jane, Rees, Jonathan, Rombach, Ines, Savulescu, Julian, Tracey, Irene, Wartolowska, Karolina, Blazeby, Jane M., Barham, Paul, Brookes, Sara T., Crosby, Tom, Falk, Stephen J., Griffin, S. Michael, Hollingworth, William, Hollowood, Andrew D., Krysztopik, Richard, Lewis, Wyn, Nicklin, Jo, Streets, Christopher, Strong, Sean, Titcomb, Dan, Williams, Geraint, Birtle, Alison, Bryan, Rik, Catto, James, Chester, John, French, Ann, Hall, Emma, Harris, Chris, Johnson, Mark, Jones, Rob, Keeley, Francis, Kirkbank, Tony, Kockelbergh, Roger, Lewis, Rebecca, Newton, Michelle, Powles, Thomas, Waters, Rachel, Winterbottom, Andrew, Halliday, Alison, Becquemin, Jean-Pierre, Belli, Anna, Bosiers, Marc, Cao, Piergiorgio, Davies, Christina, Gough, Michael, Hayter, Elizabeth, Leopold, Peter, McDonald, Sumaira, Michaels, Jonathan, Mihaylova, Borislava, Peto, Richard, Robertson, Steven, Rothwell, Peter, Scott, Rachael, Thomas, Dafydd, Vermassen, Frank, Stein, Rob, Bartlett, John, Cameron, David, Campbell, Amy, Canney, Peter, Dunn, Janet, Earl, Helena, Falzon, Mary, Francis, Adele, Hall, Peter, Harmer, Victoria, Higgins, Helen, Hiller, Louise, Hughes-Davies, Luke, Macpherson, Iain, Makris, Andreas, Marshall, Andrea, McCabe, Christopher, Morgan, Adrienne, Pinder, Sarah, Poole, Christopher, Rea, Daniel, Stallard, Nigel

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