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Search Results - Okumura-Kitajima, Lisa
Search Results - Okumura-Kitajima, Lisa
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Design, synthesis and biological evaluation of novel pyridine derivatives as gut-selective NaPi2b inhibitors
by
Ushiki, Yasunobu
,
Kawabe, Kenichi
,
Yamamoto-Okada, Kumiko
,
Uneuchi, Fumito
,
Asanuma, Yuta
,
Yamaguchi, Chitose
,
Ohta, Hiroshi
,
Shibata, Tsuyoshi
,
Abe, Tomohiro
,
Okumura-Kitajima, Lisa
,
Kosai, Yuki
,
Endo, Mayumi
,
Otake, Katsumasa
,
Munetomo, Eiji
,
Takahashi, Teisuke
,
Kakinuma, Hiroyuki
Published in
Bioorganic & medicinal chemistry letters
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Design, synthesis and biological evaluation of novel indole derivatives as gut-selective NaPi2b inhibitors
by
Ushiki, Yasunobu
,
Kawabe, Kenichi
,
Yamamoto-Okada, Kumiko
,
Uneuchi, Fumito
,
Asanuma, Yuta
,
Yamaguchi, Chitose
,
Ohta, Hiroshi
,
Shibata, Tsuyoshi
,
Abe, Tomohiro
,
Okumura-Kitajima, Lisa
,
Kosai, Yuki
,
Endo, Mayumi
,
Otake, Katsumasa
,
Munetomo, Eiji
,
Takahashi, Teisuke
,
Kakinuma, Hiroyuki
Published in
Bioorganic & medicinal chemistry
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(1S)-1,5-Anhydro-1-[5-(4-ethoxybenzyl)-2-methoxy-4-methylphenyl]-1-thio-d-glucitol (TS-071) is a Potent, Selective Sodium-Dependent Glucose Cotransporter 2 (SGLT2) Inhibitor for Ty...
by
Kakinuma, Hiroyuki
,
Oi, Takahiro
,
Hashimoto-Tsuchiya, Yuko
,
Arai, Masayuki
,
Kawakita, Yasunori
,
Fukasawa, Yoshiki
,
Iida, Izumi
,
Hagima, Naoko
,
Takeuchi, Hiroyuki
,
Chino, Yukihiro
,
Asami, Jun
,
Okumura-Kitajima, Lisa
,
Io, Fusayo
,
Yamamoto, Daisuke
,
Miyata, Noriyuki
,
Takahashi, Teisuke
,
Uchida, Saeko
,
Yamamoto, Koji
Published in
Journal of medicinal chemistry
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Discovery of potent, low-absorbable sodium-dependent glucose cotransporter 1 (SGLT1) inhibitor SGL5213 for type 2 diabetes treatment
by
Kuroda, Shoichi
,
Kobashi, Yohei
,
Oi, Takahiro
,
Kawabe, Kenichi
,
Shiozawa, Fumiyasu
,
Okumura-Kitajima, Lisa
,
Sugisaki-Kitano, Mami
,
Io, Fusayo
,
Yamamoto, Koji
,
Kakinuma, Hiroyuki
Published in
Bioorganic & medicinal chemistry
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Design, synthesis and biological evaluation of novel 1H-pyrazole-4-carbonyl-4,5,6,7-tetrahydrobenzo [b]thiophene derivatives as gut-selective NaPi2b inhibitors
by
Ushiki, Yasunobu
,
Kawabe, Kenichi
,
Yamamoto-Okada, Kumiko
,
Uneuchi, Fumito
,
Asanuma, Yuta
,
Yamaguchi, Chitose
,
Ohta, Hiroshi
,
Shibata, Tsuyoshi
,
Abe, Tomohiro
,
Okumura-Kitajima, Lisa
,
Kosai, Yuki
,
Endo, Mayumi
,
Otake, Katsumasa
,
Munetomo, Eiji
,
Takahashi, Teisuke
,
Kakinuma, Hiroyuki
Published in
Bioorganic & medicinal chemistry letters
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Discovery of a potent, low-absorbable sodium-dependent glucose cotransporter 1 (SGLT1) inhibitor (TP0438836) for the treatment of type 2 diabetes
by
Kuroda, Shoichi
,
Kobashi, Yohei
,
Oi, Takahiro
,
Amada, Hideaki
,
Okumura-Kitajima, Lisa
,
Io, Fusayo
,
Yamamto, Koji
,
Kakinuma, Hiroyuki
Published in
Bioorganic & medicinal chemistry letters
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Discovery of novel 2-[(4-hydroxy-6-oxo-2,3-dihydro-1H-pyridine-5-carbonyl)amino]acetic acid derivatives as HIF prolyl hydroxylase inhibitors for treatment of renal anemia
by
Hamada, Makoto
,
Takayama, Tetsuo
,
Shibata, Tsuyoshi
,
Hiratate, Akira
,
Takahashi, Masato
,
Yashiro, Miyoko
,
Takayama, Noriko
,
Okumura-Kitajima, Lisa
,
Koretsune, Hiroko
,
Kajiyama, Hiromitsu
,
Naruse, Takumi
,
Kato, Sota
,
Takano, Hiroki
,
Kakinuma, Hiroyuki
Published in
Bioorganic & medicinal chemistry letters
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Lead generation from N-[benzyl(4-phenylbutyl)carbamoyl]amino acid as a novel LPA1 antagonist for the treatment of systemic sclerosis
by
Kobayashi, Yuki
,
Uneuchi, Fumito
,
Naruse, Takumi
,
Matsuda, Daisuke
,
Okumura-Kitajima, Lisa
,
Kajiyama, Hiromitsu
,
Wada, Reiko
,
Yonemoto, Yuki
,
Nakano, Koichiro
,
Toki, Hidetoh
,
Kamigaso, Shunsuke
,
Yamagishi, Jyunya
,
Tokura, Seiken
,
Kakinuma, Hiroyuki
,
Kuroda, Shoichi
Published in
European journal of medicinal chemistry
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Lead generation from N-benzyl(4-phenylbutyl)carbamoylamino acid as a novel LPA1 antagonist for the treatment of systemic sclerosis
by
Kobayashi, Yuki
,
Uneuchi, Fumito
,
Naruse, Takumi
,
Matsuda, Daisuke
,
Okumura-Kitajima, Lisa
,
Kajiyama, Hiromitsu
,
Wada, Reiko
,
Yonemoto, Yuki
,
Nakano, Koichiro
,
Toki, Hidetoh
,
Kamigaso, Shunsuke
,
Yamagishi, Jyunya
,
Tokura, Seiken
,
Kakinuma, Hiroyuki
,
Kuroda, Shoichi
Published in
European journal of medicinal chemistry
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SGL5213, a novel and potent intestinal SGLT1 inhibitor, suppresses intestinal glucose absorption and enhances plasma GLP-1 and GLP-2 secretion in rats
by
Io, Fusayo
,
Gunji, Emi
,
Koretsune, Hiroko
,
Kato, Koji
,
Sugisaki-Kitano, Mami
,
Okumura-Kitajima, Lisa
,
Kimura, Kayo
,
Uchida, Saeko
,
Yamamoto, Koji
Published in
European journal of pharmacology
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(2 S,4 S)-4-Fluoro-1-{[(2-hydroxy-1,1-dimethylethyl)amino]acetyl}-pyrrolidine-2-carbonitrile monobenzenesulfonate (TS-021) is a selective and reversible dipeptidyl peptidase IV inh...
by
Tajima, Atsushi
,
Yamamoto, Koji
,
Kozakai, Akinori
,
Okumura-Kitajima, Lisa
,
Mita, Yasuo
,
Kitano, Kiyokazu
,
Jingu, Shigeji
,
Nakaike, Shiro
Published in
European journal of pharmacology
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