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Structure-based design and modular synthesis of novel PI4K class II inhibitors bearing a 4-aminoquinazoline scaffold
by
Misehe, Mbilo
,
Klima, Martin
,
Matoušová, Marika
,
Chalupská, Dominika
,
Dejmek, Milan
,
Šála, Michal
,
Mertlíková-Kaiserová, Helena
,
Boura, Evzen
,
Nencka, Radim
Published in
Bioorganic & medicinal chemistry letters
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Design, synthesis and evaluation of novel thieno[2,3d]pyrimidine derivatives as potent and specific RIPK2 inhibitors
by
Misehe, Mbilo
,
Šála, Michal
,
Matoušová, Marika
,
Hercík, Kamil
,
Kocek, Hugo
,
Chalupská, Dominika
,
Chaloupecká, Ema
,
Hájek, Miroslav
,
Boura, Evzen
,
Mertlíková-Kaiserová, Helena
,
Nencka, Radim
Published in
Bioorganic & medicinal chemistry letters
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1,2,4-Thiadiazole acyclic nucleoside phosphonates as inhibitors of cysteine dependent enzymes cathepsin K and GSK-3β
by
Pomeislová, Alice
,
Otmar, Miroslav
,
Rubešová, Petra
,
Benýšek, Jakub
,
Matoušová, Marika
,
Mertlíková-Kaiserová, Helena
,
Pohl, Radek
,
Poštová Slavětínská, Lenka
,
Pomeisl, Karel
,
Krečmerová, Marcela
Published in
Bioorganic & medicinal chemistry
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Structurally Redesigned Bioorthogonal Reagents for Mitochondria-Specific Prodrug Activation
by
Dzijak, Rastislav
,
Galeta, Juraj
,
Vázquez, Arcadio
,
Kozák, Jaroslav
,
Matoušová, Marika
,
Fulka, Helena
,
Dračínský, Martin
,
Vrabel, Milan
Published in
JACS Au
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Role of Caspases and CD95/Fas in the Apoptotic Effects of a Nucleotide Analog PMEG in CCRF-CEM Cells
by
MERTLIKOVA-KAISEROVA, Helena
,
VOTRUBA, Ivan
,
MATOUSOVA, Marika
,
HOLY, Antonín
,
HAJEK, Miroslav
Published in
Anticancer research
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Rational Design of Novel Highly Potent and Selective Phosphatidylinositol 4‑Kinase IIIβ (PI4KB) Inhibitors as Broad-Spectrum Antiviral Agents and Tools for Chemical Biology
by
Mejdrová, Ivana
,
Chalupská, Dominika
,
Plačková, Pavla
,
Müller, Christin
,
Šála, Michal
,
Klíma, Martin
,
Baumlová, Adriana
,
Hřebabecký, Hubert
,
Procházková, Eliška
,
Dejmek, Milan
,
Strunin, Dmytro
,
Weber, Jan
,
Lee, Gary
,
Matoušová, Marika
,
Mertlíková-Kaiserová, Helena
,
Ziebuhr, John
,
Birkus, Gabriel
,
Boura, Evzen
,
Nencka, Radim
Published in
Journal of medicinal chemistry
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Fluorescent Inhibitors as Tools To Characterize Enzymes: Case Study of the Lipid Kinase Phosphatidylinositol 4‑Kinase IIIβ (PI4KB)
by
Humpolickova, Jana
,
Mejdrová, Ivana
,
Matousova, Marika
,
Nencka, Radim
,
Boura, Evzen
Published in
Journal of medicinal chemistry
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Synthesis of sulfur karrikin bioisosteres as potential neuroprotectives
by
Pošta, Martin
,
Zima, Václav
,
Poštová Slavětínská, Lenka
,
Matoušová, Marika
,
Beier, Petr
Published in
Beilstein journal of organic chemistry
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Pregn-5-en-3β-ol and androst-5-en-3β-ol dicarboxylic acid esters as potential therapeutics for NMDA hypofunction: In vitro safety assessment and plasma stability
by
Matousova, Marika
,
Soucek, Radko
,
Tloustova, Eva
,
Slavikova, Barbora
,
Chodounska, Hana
,
Mertlikova-Kaiserova, Helena
,
Kudova, Eva
Published in
Steroids
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Screening of novel 3α5β-neurosteroids for neuroprotective activity against glutamate- or NMDA-induced excitotoxicity
by
Smidkova, Marketa
,
Hajek, Miroslav
,
Adla, Santosh Kumar
,
Slavikova, Barbora
,
Chodounska, Hana
,
Matousova, Marika
,
Mertlikova-Kaiserova, Helena
,
Kudova, Eva
Published in
The Journal of steroid biochemistry and molecular biology
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Fluorescence‐Based HTS Assays for Ion Channel Modulation in Drug Discovery Pipelines
by
Voldřich, Jan
,
Matoušová, Marika
,
Šmídková, Markéta
,
Mertlikova-Kaiserova, Helena
Published in
ChemMedChem
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Identification of N-methyl-D-aspartate receptor antagonists using the rat postnatal mixed cortical and hippocampal neurons
by
Voldřich, Jan
,
Matoušová, Marika
,
Šmídková, Markéta
,
Slavíková, Barbora
,
Chodounská, Hana
,
Kudová, Eva
,
Mertlíková-Kaiserová, Helena
Published in
European journal of pharmacology
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