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Discovery of SAR184841, a potent and long-lasting inhibitor of 11β-hydroxysteroid dehydrogenase type 1, active in a physiopathological animal model of T2D
by
Venier, Olivier
,
Pascal, Cécile
,
Braun, Alain
,
Namane, Claudie
,
Mougenot, Patrick
,
Crespin, Olivier
,
Pacquet, François
,
Mougenot, Cécile
,
Monseau, Catherine
,
Onofri, Bénédicte
,
Dadji-Faïhun, Rommel
,
Leger, Céline
,
Ben-Hassine, Majdi
,
Van-Pham, Thao
,
Ragot, Jean-Luc
,
Philippo, Christophe
,
Farjot, Géraldine
,
Noah, Lionel
,
Maniani, Karima
,
Boutarfa, Asma
,
Nicolaï, Eric
,
Guillot, Etienne
,
Pruniaux, Marie-Pierre
,
Güssregen, Stefan
,
Engel, Christian
,
Coutant, Anne-Laure
,
de Miguel, Beatriz
,
Castro, Antonio
Published in
Bioorganic & medicinal chemistry letters
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Pyrrolidine-pyrazole ureas as potent and selective inhibitors of 11β-hydroxysteroid-dehydrogenase type 1
by
Venier, Olivier
,
Pascal, Cécile
,
Braun, Alain
,
Namane, Claudie
,
Mougenot, Patrick
,
Crespin, Olivier
,
Pacquet, François
,
Mougenot, Cécile
,
Monseau, Catherine
,
Onofri, Bénédicte
,
Dadji-Faïhun, Rommel
,
Leger, Céline
,
Ben-Hassine, Majdi
,
Van-Pham, Thao
,
Ragot, Jean-Luc
,
Philippo, Christophe
,
Güssregen, Stefan
,
Engel, Christian
,
Farjot, Géraldine
,
Noah, Lionel
,
Maniani, Karima
,
Nicolaï, Eric
Published in
Bioorganic & medicinal chemistry letters
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Discovery of SAR184841, a potent and long-lasting inhibitor of 11[beta]-hydroxysteroid dehydrogenase type 1, active in a physiopathological animal model of T2D
by
Venier, Olivier
,
Pascal, Cecile
,
Braun, Alain
,
Namane, Claudie
,
Mougenot, Patrick
,
Crespin, Olivier
,
Pacquet, Francois
,
Mougenot, Cecile
,
Monseau, Catherine
,
Onofri, Benedicte
,
Dadji-Faiehun, Rommel
,
Leger, Celine
,
Ben-Hassine, Majdi
,
Van-Pham, Thao
,
Ragot, Jean-Luc
,
Philippo, Christophe
,
Farjot, Geraldine
,
Noah, Lionel
,
Maniani, Karima
,
Boutarfa, Asma
,
Nicolaie, Eric
,
Guillot, Etienne
,
Pruniaux, Marie-Pierre
,
Guessregen, Stefan
,
Engel, Christian
,
Coutant, Anne-Laure
,
de Miguel, Beatriz
,
Castro, Antonio
Published in
Bioorganic & medicinal chemistry letters
Get full text
Article
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Bioorganic & Medicinal Chemistry Letters
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Subjects
11-Beta-Hydroxysteroid Dehydrogenase Type 1 - Antagonists & Inhibitors
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2
11-Beta-Hydroxysteroid Dehydrogenase Type 1 - Metabolism
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2
Animals
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Chemistry
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Chemistry, Medicinal
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Chemistry, Organic
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Humans
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Life Sciences & Biomedicine
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Metabolic Syndrome
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Mice
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Pharmacodynamic Ex Vivo Assay
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Pharmacology & Pharmacy
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Physical Sciences
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Science & Technology
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11Β-Hsd-1 Inhibitors
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1
11Β-Hsd1 Inhibitors
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1
11Β-Hydroxysteroid-Dehydrogenase Type 1
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1
11Β-Hydroxysteroid-Dehydrogenase Type I
1 results
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Adamantane - Chemistry
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1
Adamantane - Pharmacokinetics
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Sciencedirect
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Sciencedirect Freedom Collection 2022-2024
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Science Citation Index Expanded (Web Of Science)
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Backfile Package - Organic Chemistry (Legacy) [Yco]
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2