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Search Results - Gunawardana, Indrani
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Spirocyclic β‑Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1) Inhibitors: From Hit to Lowering of Cerebrospinal Fluid (CSF) Amyloid β in a Higher Species
by
Hunt, Kevin W
,
Cook, Adam W
,
Watts, Ryan J
,
Clark, Christopher T
,
Vigers, Guy
,
Smith, Darin
,
Metcalf, Andrew T
,
Gunawardana, Indrani W
,
Burkard, Michael
,
Cox, April A
,
Geck Do, Mary K
,
Dutcher, Darrin
,
Thomas, Allen A
,
Rana, Sumeet
,
Kallan, Nicholas C
,
DeLisle, Robert K
,
Rizzi, James P
,
Regal, Kelly
,
Sammond, Douglas
,
Groneberg, Robert
,
Siu, Michael
,
Purkey, Hans
,
Lyssikatos, Joseph P
,
Marlow, Allison
,
Liu, Xingrong
,
Tang, Tony P
Published in
Journal of medicinal chemistry
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Discovery of 7‑Tetrahydropyran-2-yl Chromans: β‑Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1) Inhibitors That Reduce Amyloid β‑Protein (Aβ) in the Central Nervous System...
by
Thomas, Allen A
,
Hunt, Kevin W
,
Volgraf, Matthew
,
Watts, Ryan J
,
Liu, Xingrong
,
Vigers, Guy
,
Smith, Darin
,
Sammond, Douglas
,
Tang, Tony P
,
Rhodes, Susan P
,
Metcalf, Andrew T
,
Brown, Karin D
,
Otten, Jennifer N
,
Burkard, Michael
,
Cox, April A
,
Do, Mary K. Geck
,
Dutcher, Darrin
,
Rana, Sumeet
,
DeLisle, Robert K
,
Regal, Kelly
,
Wright, Albion D
,
Groneberg, Robert
,
Scearce-Levie, Kimberly
,
Siu, Michael
,
Purkey, Hans E
,
Lyssikatos, Joseph P
,
Gunawardana, Indrani W
Published in
Journal of medicinal chemistry
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Selective Inhibition of ICAM-1 and E-Selectin Expression in Human Endothelial Cells. 2. Aryl Modifications of 4-(Aryloxy)thieno[2,3-c]pyridines with Fine-Tuning at C-2 Carbamides
by
Zhu, Gui-Dong
,
Arendsen, David L
,
Gunawardana, Indrani W
,
Boyd, Steven A
,
Stewart, Andrew O
,
Fry, Dennis G
,
Cool, Barbara L
,
Kifle, Lemma
,
Schaefer, Verlyn
,
Meuth, Joseph
,
Marsh, Kennan C
,
Kempf-Grote, Anita J
,
Kilgannon, Patrick
,
Gallatin, W. Michael
,
Okasinski, Gregory F
Published in
Journal of medicinal chemistry
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Discovery of Inhibitors of Cell Adhesion Molecule Expression in Human Endothelial Cells. 1. Selective Inhibition of ICAM-1 and E-Selectin Expression
by
Stewart, Andrew O
,
Bhatia, Pramila A
,
McCarty, Catherine M
,
Patel, Meena V
,
Staeger, Michael A
,
Arendsen, David L
,
Gunawardana, Indrani W
,
Melcher, Laura M
,
Zhu, Gui-Dong
,
Boyd, Steven A
,
Fry, Dennis G
,
Cool, Barbara L
,
Kifle, Lemma
,
Lartey, Kraig
,
Marsh, Kennan C
,
Kempf-Grote, Anita J
,
Kilgannon, Patrick
,
Wisdom, Wendy
,
Meyer, Joey
,
Gallatin, W. Michael
,
Okasinski, Gregory F
Published in
Journal of medicinal chemistry
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Non-charged thiamine analogs as inhibitors of enzyme transketolase
by
Thomas, Allen A.
,
De Meese, J.
,
Le Huerou, Y.
,
Boyd, Steven A.
,
Romoff, Todd T.
,
Gonzales, Steven S.
,
Gunawardana, Indrani
,
Kaplan, Tomas
,
Sullivan, Francis
,
Condroski, Kevin
,
Lyssikatos, Joseph P.
,
Aicher, Thomas D.
,
Ballard, Josh
,
Bernat, Bryan
,
DeWolf, Walter
,
Han, May
,
Lemieux, Christine
,
Smith, Darin
,
Weiler, Solly
,
Wright, S. Kirk
,
Vigers, Guy
,
Brandhuber, Barb
Published in
Bioorganic & medicinal chemistry
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Abstract 3874: Single-agent Chk1 inhibition is anti-proliferative in leukemia cells in vitro and in vivo
by
Davies, Kurtis D.
,
Humphries, Michael J.
,
Sullivan, Francis
,
von Carlowitz, Ira
,
Huerou, Yvan Le
,
Mohr, Peter J.
,
Wang, Bin
,
Blake, Jim F.
,
Lyon, Michael A.
,
Gunawardana, Indrani
,
Chicarelli, Mark
,
Wallace, Eli
,
Gross, Stefan
Published in
Cancer research (Chicago, Ill.)
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Prodrug thiamine analogs as inhibitors of the enzyme transketolase
by
Le Huerou, Yvan
,
Gunawardana, Indrani
,
Thomas, Allen A.
,
Boyd, Steven A.
,
de Meese, Jason
,
deWolf, Walter
,
Gonzales, Steven S.
,
Han, May
,
Hayter, Laura
,
Kaplan, Tomas
,
Lemieux, Christine
,
Lee, Patrice
,
Pheneger, Jed
,
Poch, Gregory
,
Romoff, Todd T.
,
Sullivan, Francis
,
Weiler, Solly
,
Wright, S. Kirk
,
Lin, Jie
Published in
Bioorganic & medicinal chemistry
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Abstract B254: Extended target-coverage by selective Chk1 inhibitors enhances pharmacodynamic inhibition of Chk1 signaling and antitumor activity in vivo
by
Humphries, Michael J.
,
von Carlowitz, Ira
,
Le Huerou, Yvan
,
Randolph, Nikole
,
Mohr, Peter J.
,
Wang, Bin
,
Lyon, Michael A.
,
Gunawardana, Indrani
,
Chicarelli, Mark
,
Blake, Jim F.
,
Schrag, Michael L.
,
Winski, Shannon L.
,
Wallace, Eli
Published in
Molecular cancer therapeutics
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New Antimitotic Agents with Activity in Multi-Drug-Resistant Cell Lines and in Vivo Efficacy in Murine Tumor Models
by
Szczepankiewicz, Bruce G
,
Liu, Gang
,
Jae, Hwan-Soo
,
Tasker, Andrew S
,
Gunawardana, Indrani W
,
von Geldern, Thomas W
,
Gwaltney, Stephen L
,
Wu-Wong, J. Ruth
,
Gehrke, Laura
,
Chiou, William J
,
Credo, R. Bruce
,
Alder, Jeffery D
,
Nukkala, Michael A
,
Zielinski, Nicolette A
,
Jarvis, Ken
,
Mollison, Karl W
,
Frost, David J
,
Bauch, Joy L
,
Hui, Yu Hua
,
Claiborne, Akiyo K
,
Li, Qun
,
Rosenberg, Saul H
Published in
Journal of medicinal chemistry
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A facile and general synthesis of 2,4-Di- and 2,4,7-trisubstituted thieno[2,3-c]pyridines
by
Zhu, Gui-Dong
,
Gunawardana, Indrani W.
,
Boyd, Steven A.
,
Melcher, Laura M.
Published in
Journal of heterocyclic chemistry
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11
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Studies on an immunosuppressive macrolactam, ascomycin: Synthesis of a C-33 hydroxyl derivative
by
Kawai, Megumi
,
Gunawardana, Indrani W.K.
,
Mollison, Karl W.
,
Hsieh, Gin C.
,
Lane, Benjamin C.
,
Luly, Jay R.
Published in
Bioorganic & medicinal chemistry letters
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