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Time-resolved FRET screening identifies small molecular modifiers of mutant Huntingtin conformational inflexibility in patient-derived cells
by
Wilbertz, Johannes H.
,
Frappier, Julia
,
Muller, Sandra
,
Gratzer, Sabine
,
Englaro, Walter
,
Stanek, Lisa M.
,
Calamini, Barbara
Published in
SLAS discovery
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Abstract 6425: Sensitivity of oncogenic KRAS-expressing cells to CDK9 inhibition identified by a phenotypic compound screen
by
Lai, Lick P.
,
Brel, Viviane
,
Sharma, Kanika
,
Frappier, Julia
,
Le-Henanf, Nadia
,
Vivet, Bertrand
,
Muzet, Nicolas
,
Schell, Emilie
,
Morales, Renaud
,
Rooney, Eamonn
,
Holderfield, Matthew
,
Lacroix, Frederic
,
Englaro, Walter
,
Marcireau, Christophe
,
Debussche, Laurent
,
Nissley, Dwight V.
,
Mccormick, Frank
Published in
Cancer research (Chicago, Ill.)
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Sensitivity of Oncogenic KRAS-Expressing Cells to CDK9 Inhibition
by
Lai, Lick Pui
,
Brel, Viviane
,
Sharma, Kanika
,
Frappier, Julia
,
Le-Henanf, Nadia
,
Vivet, Bertrand
,
Muzet, Nicolas
,
Schell, Emilie
,
Morales, Renaud
,
Rooney, Eamonn
,
Basse, Nicolas
,
Yi, Ming
,
Lacroix, Frederic
,
Holderfield, Matthew
,
Englaro, Walter
,
Marcireau, Christophe
,
Debussche, Laurent
,
Nissley, Dwight V.
,
McCormick, Frank
Published in
SLAS discovery
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Slas Discovery
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Cancer Research
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Biochemical Research Methods
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Cdk9
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Cyclin-Dependent Kinase 9 - Antagonists & Inhibitors
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Drug Discovery - Methods
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Drug Screening Assays, Antitumor - Methods
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Gene Expression Regulation, Neoplastic - Drug Effects
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High-Throughput Screening Assays
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