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Identification of a Chemical Probe for Bromo and Extra C‑Terminal Bromodomain Inhibition through Optimization of a Fragment-Derived Hit
by
Fish, Paul V
,
Filippakopoulos, Panagis
,
Bish, Gerwyn
,
Brennan, Paul E
,
Bunnage, Mark E
,
Cook, Andrew S
,
Federov, Oleg
,
Gerstenberger, Brian S
,
Jones, Hannah
,
Knapp, Stefan
,
Marsden, Brian
,
Nocka, Karl
,
Owen, Dafydd R
,
Philpott, Martin
,
Picaud, Sarah
,
Primiano, Michael J
,
Ralph, Michael J
,
Sciammetta, Nunzio
,
Trzupek, John D
Published in
Journal of medicinal chemistry
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SARS-CoV-2 infects the human kidney and drives fibrosis in kidney organoids
by
Reimer, Katharina C.
,
Nagai, James S.
,
Varghese, Finny S.
,
Overheul, Gijs J.
,
Roverts, Rona
,
Willemsen, Brigith
,
Beukenboom, Marcel
,
Dunnen, Wilfred den
,
Triana, Sergio H.
,
Timm, Marie-Cherelle
,
van den Berge, Bartholomeus T.
,
Nlandu, Quincy
,
Heijnert, Joelle
,
Bindels, Eric M.J.
,
Hoogenboezem, Remco M.
,
Mooren, Fieke
,
Kuppe, Christoph
,
Grünberg, Katrien
,
Steenbergen, Eric J.
,
Czogalla, Jan
,
Sommerdijk, Nico
,
Akiva, Anat
,
Boor, Peter
,
Huber, Tobias B.
,
Bar-David, Elad
,
Barr, Haim
,
Boby, Melissa L.
,
Borden, Bruce
,
Bowman, Gregory R.
,
Brun, Juliane
,
BVNBS, Sarma
,
Carbery, Anna
,
Chernychenko, Eugene
,
Clyde, Austin
,
Coffland, Joseph E.
,
Cole, Jason
,
Cox, Lisa
,
Dudgeon, Tim
,
Dunnett, Louise
,
Erez, Noam
,
Fate, Gwen
,
Ferrins, Lori
,
Foster, Richard
,
Foster, Holly
,
Gabizon, Ronen
,
Gawriljuk, Victor O.
,
Gehrtz, Paul
,
Gileadi, Carina
,
Giroud, Charline
,
Glen, Robert
,
Gorichko, Marian
,
Griffen, Ed J.
,
Heer, Jag
,
Hill, Michelle
,
Horrell, Sam
,
Jajack, Andrew
,
De Jonghe, Steven
,
Kantsadi, Anastassia L.
,
Koekemoer, Lizbe
,
Lee, Alpha A.
,
Lefker, Bruce A.
,
Macdonald, Hannah Bruce
,
Maclean, Beth
,
McCorkindale, Willam
,
McGovern, Briana L.
,
Michurin, Oleg
,
Morris, Aaron
,
Morris, Garret M.
,
Neyts, Johan
,
Oliva, Glaucius
,
Overheul, Gijs J.
,
Owen, David
,
Psenak, Vladimir
,
Pai, Ruby
,
Paran, Nir
,
Perry, Benjamin
,
Pingle, Maneesh
,
Politi, Boaz
,
Powell, Ailsa
,
Puni, Reut
,
Resnick, Efrat
,
Rosales, Romel
,
Schofield, Chris
,
Shafeev, Mikhail
,
Sittner, Assa
,
Skyner, Rachael
,
Spencer, John
,
Tamir, Hadas
,
Tennant, Rachael
,
Tumber, Anthony
,
van Rij, Ronald P.
,
Voelz, Vincent
,
Volkamer, Andra
,
von Delft, Annette
,
White, Kris M.
,
Wright, Nathan
,
Zidane, Hadeer
,
Costa, Ivan G.
,
Schneider, Rebekka K.
,
Smeets, Bart
Published in
Cell stem cell
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Sulfated Glycosaminoglycans Control the Extracellular Trafficking and the Activity of the Metalloprotease Inhibitor TIMP-3
by
Troeberg, Linda
,
Lazenbatt, Christopher
,
Anower-E-Khuda, Md. Ferdous
,
Freeman, Craig
,
Federov, Oleg
,
Habuchi, Hiroko
,
Habuchi, Osami
,
Kimata, Koji
,
Nagase, Hideaki
Published in
Chemistry & biology
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Abstract 5084: Potent and isoform-selective ATAD2 bromodomain inhibitor with unprecedented chemical structure and mode of action
by
Fernández-Montalván, Amaury E.
,
Berger, Markus
,
Kuropka, Benno
,
Koo, Seong Joo
,
Badock, Volker
,
Weiske, Joerg
,
Holton, Simon J.
,
Chaikuad, Apirat
,
Díaz-Sáez, Laura
,
Bennett, James
,
Federov, Oleg
,
Huber, Kilian
,
Centrella, Paolo
,
Clark, Matthew A.
,
Dumelin, Christoph E.
,
Sigel, Eric A.
,
Soutter, Holly S.
,
Troast, Dawn M.
,
Zhang, Ying
,
Cuozzo, John W.
,
Keefe, Anthony D.
,
Roche, Didier
,
Rodeschini, Vincent
,
Hübner, Jan
,
Weinmann, Hilmar
,
Hartung, Ingo V.
,
Gorjanacz, Matyas
Published in
Cancer research (Chicago, Ill.)
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Taking Stock: Documenting Russia's Modern Heritage
by
Anderson, Richard
Published in
Future Anterior: Journal of Historic Preservation, History, Theory, and Criticism
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