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Search Results - Ellis-Hutchings, Michelle
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Evaluation of farnesyl:Protein transferase and geranylgeranyl:Protein transferase inhibitor combinations in preclinical models
by
LOBELL, Robert B
,
OMER, Charles A
,
KRAL, Astrid M
,
DONGMING LIU
,
LUMMA, William C
,
MACHOTKA, Samuel V
,
RANDS, Elaine
,
WILLIAMS, Theresa M
,
GRAHAM, Samuel L
,
HARTMAN, George D
,
OLIFF, Allen I
,
HEIMBROOK, David C
,
ABRAMS, Marc T
,
KOHL, Nancy E
,
BHIMNATHWALA, Hema G
,
BRUCKER, Mary Jo
,
BUSER, Carolyn A
,
DAVIDE, Joseph P
,
DESOLMS, S. Jane
,
DINSMORE, Christopher J
,
ELLIS-HUTCHINGS, Michelle S
Published in
Cancer research (Chicago, Ill.)
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The synthesis and biological evaluation of a series of potent dual inhibitors of farnesyl and geranyl-Geranyl protein transferases
by
Tucker, Thomas J
,
Abrams, Marc T
,
Buser, Carolyn A
,
Davide, Joseph P
,
Ellis-Hutchings, Michelle
,
Fernandes, Christine
,
Gibbs, Jackson B
,
Graham, Samuel L
,
Hartman, George D
,
Huber, Hans E
,
Liu, Dongming
,
Lobell, Robert B
,
Lumma, William C
,
Robinson, Ronald G
,
Sisko, John T
,
Smith, Anthony M
Published in
Bioorganic & medicinal chemistry letters
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3-Aminopyrrolidinone Farnesyltransferase Inhibitors: Design of Macrocyclic Compounds with Improved Pharmacokinetics and Excellent Cell Potency
by
Bell, Ian M
,
Gallicchio, Steven N
,
Abrams, Marc
,
Beese, Lorena S
,
Beshore, Douglas C
,
Bhimnathwala, Hema
,
Bogusky, Michael J
,
Buser, Carolyn A
,
Culberson, J. Christopher
,
Davide, Joseph
,
Ellis-Hutchings, Michelle
,
Fernandes, Christine
,
Gibbs, Jackson B
,
Graham, Samuel L
,
Hamilton, Kelly A
,
Hartman, George D
,
Heimbrook, David C
,
Homnick, Carl F
,
Huber, Hans E
,
Huff, Joel R
,
Kassahun, Kelem
,
Koblan, Kenneth S
,
Kohl, Nancy E
,
Lobell, Robert B
,
Lynch, Joseph J
,
Robinson, Ronald
,
Rodrigues, A. David
,
Taylor, Jeffrey S
,
Walsh, Eileen S
,
Williams, Theresa M
,
Zartman, C. Blair
Published in
Journal of medicinal chemistry
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Dual Protein Farnesyltransferase−Geranylgeranyltransferase-I Inhibitors as Potential Cancer Chemotherapeutic Agents
by
deSolms, S. Jane
,
Ciccarone, Terrence M
,
MacTough, Suzanne C
,
Shaw, Anthony W
,
Buser, Carolyn A
,
Ellis-Hutchings, Michelle
,
Fernandes, Christine
,
Hamilton, Kelly A
,
Huber, Hans E
,
Kohl, Nancy E
,
Lobell, Robert B
,
Robinson, Ronald G
,
Tsou, Nancy N
,
Walsh, Eileen S
,
Graham, Samuel L
,
Beese, Lorena S
,
Taylor, Jeffrey S
Published in
Journal of medicinal chemistry
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Design and Biological Activity of (S)-4-(5-{[1-(3-Chlorobenzyl)-2- oxopyrrolidin-3-ylamino]methyl}imidazol-1-ylmethyl)benzonitrile, a 3-Aminopyrrolidinone Farnesyltransferase Inhib...
by
Bell, Ian M
,
Gallicchio, Steven N
,
Abrams, Marc
,
Beshore, Douglas C
,
Buser, Carolyn A
,
Culberson, J. Christopher
,
Davide, Joseph
,
Ellis-Hutchings, Michelle
,
Fernandes, Christine
,
Gibbs, Jackson B
,
Graham, Samuel L
,
Hartman, George D
,
Heimbrook, David C
,
Homnick, Carl F
,
Huff, Joel R
,
Kassahun, Kelem
,
Koblan, Kenneth S
,
Kohl, Nancy E
,
Lobell, Robert B
,
Lynch, Joseph J
,
Miller, Patricia A
,
Omer, Charles A
,
Rodrigues, A. David
,
Walsh, Eileen S
,
Williams, Theresa M
Published in
Journal of medicinal chemistry
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Potent inhibitors of farnesyltransferase and geranylgeranyltransferase-I
by
Nguyen, Diem N.
,
Stump, Craig A.
,
Walsh, Eileen S.
,
Fernandes, Christine
,
Davide, Joseph P.
,
Ellis-Hutchings, Michelle
,
Robinson, Ronald G.
,
Williams, Theresa M.
,
Lobell, Robert B.
,
Huber, Hans E.
,
Buser, Carolyn A.
Published in
Bioorganic & medicinal chemistry letters
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Macrocyclic piperazinones as potent dual inhibitors of farnesyltransferase and geranylgeranyltransferase-I
by
Dinsmore, Christopher J
,
Zartman, C.Blair
,
Bergman, Jeffrey M
,
Abrams, Marc T
,
Buser, Carolyn A
,
Culberson, J.Christopher
,
Davide, Joseph P
,
Ellis-Hutchings, Michelle
,
Fernandes, Christine
,
Graham, Samuel L
,
Hartman, George D
,
Huber, Hans E
,
Lobell, Robert B
,
Mosser, Scott D
,
Robinson, Ronald G
,
Williams, Theresa M
Published in
Bioorganic & medicinal chemistry letters
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Evaluation of amino acid-based linkers in potent macrocyclic inhibitors of farnesyl-protein transferase
by
BESHORE, Douglas C
,
BELL, Ian M
,
DAVIDE, Joseph P
,
ELLIS-HUTEHINGS, Michelle S
,
HUBER, Hans A
,
KOBLAN, Kenneth S
,
BUSER, Carolyn A
,
KOHL, Nancy E
,
LOBELL, Robert B
,
CHEN, I-Wu
,
MCLOUGHLIN, Debra A
,
OLAH, Timothy V
,
DINSMORE, Christopher J
,
GRAHAM, Samuel L
,
HARTMAN, George D
,
WILLIAMS, Theresa M
,
HOMNICK, Carl F
,
CULBERSON, J. Christopher
,
ROBINSON, Ronald G
,
FERNANDES, Christine
,
WALSH, Eileen S
,
ABRAMS, Marc T
,
BHIMNATHWALA, Hema G
Published in
Bioorganic & medicinal chemistry letters
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Design and biological activity of (S)-4-(5-{[1-(3-chlorobenzyl)-2-oxopyrrolidin-3-ylamino]methyl}imidazol-1-ylmeth yl)benzonitrile, a 3-aminopyrrolidinone farnesyltransferase inhib...
by
BELL, Ian M
,
GALLICCHIO, Steven N
,
GRAHAM, Samuel L
,
HARTMAN, George D
,
HEIMBROOK, David C
,
HOMNICK, Carl F
,
HUFF, Joel R
,
KASSAHUN, Kelem
,
KOBLAN, Kenneth S
,
KOHL, Nancy E
,
LOBELL, Robert B
,
LYNCH, Joseph J
,
ABRAMS, Marc
,
MILLER, Patricia A
,
OMER, Charles A
,
RODRIGUES, A. David
,
WALSH, Eileen S
,
WILLIAMS, Theresa M
,
BESHORE, Douglas C
,
BUSER, Carolyn A
,
CULBERSON, J. Christopher
,
DAVIDE, Joseph
,
ELLIS-HUTCHINGS, Michelle
,
FERNANDES, Christine
,
GIBBS, Jackson B
Published in
Journal of medicinal chemistry
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