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Search Results - Cuoco, Caroline A
Search Results - Cuoco, Caroline A
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Pharmacological Characterization of the Imipridone Anticancer Drug ONC201 Reveals a Negative Allosteric Mechanism of Action at the D2 Dopamine Receptor
by
Free, R Benjamin
,
Cuoco, Caroline A
,
Xie, Bing
,
Namkung, Yoon
,
Prabhu, Varun V
,
Willette, Blair K A
,
Day, Marilyn M
,
Sanchez-Soto, Marta
,
Lane, J Robert
,
Laporte, Stéphane A
,
Shi, Lei
,
Allen, Joshua E
,
Sibley, David R
Published in
Molecular pharmacology
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Pharmacological Characterization of the Imipridone Anticancer Drug ONC201 Reveals a Negative Allosteric Mechanism of Action at the D 2 Dopamine Receptor
by
Free, R. Benjamin
,
Cuoco, Caroline A.
,
Xie, Bing
,
Namkung, Yoon
,
Prabhu, Varun V.
,
Willette, Blair K.A.
,
Day, Marilyn M.
,
Sanchez-Soto, Marta
,
Lane, J. Robert
,
Laporte, Stéphane A.
,
Shi, Lei
,
Allen, Joshua E.
,
Sibley, David R.
Published in
Molecular pharmacology
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Characterization of the novel anti‐cancer therapeutic ONC201 and related analogs as non‐competitive antagonists of the D 2 dopamine receptor
by
Cuoco, Caroline A.
,
Free, R. Benjamin
,
Willette, Blair K.
,
Day, Marilyn M.
,
Lane, J. Robert
,
Allen, Joshua E.
,
Sibley, David R.
Published in
The FASEB journal
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Characterization of the novel anti‐cancer therapeutic ONC201 and related analogs as non‐competitive antagonists of the D2 dopamine receptor
by
Cuoco, Caroline A.
,
Free, R. Benjamin
,
Willette, Blair K.
,
Day, Marilyn M.
,
Lane, J. Robert
,
Allen, Joshua E.
,
Sibley, David R.
Published in
The FASEB journal
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Abstract 5688: IND-enabling characterization of ONC206 as the next bitopic antagonist for oncology
by
Prabhu, Varun Vijay
,
Morrow, Sara
,
Cuoco, Caroline A.
,
Kawakibi, Abed R.
,
Jung, Jinkyu
,
Madhukar, Neel
,
Garnett, Matthew J.
,
McDermott, Ultan
,
Benes, Cyril H.
,
Wechsler-Reya, Robert
,
Anantharaman, Lakshmi
,
Charter, Neil
,
Rucker, Joseph B.
,
Doranz, Benjamin J.
,
Basken, Joel
,
Elemento, Olivier
,
Free, R. Benjamin
,
Sibley, David R.
,
Stogniew, Martin
,
Oster, Wolfgang
,
Gilbert, Mark R.
,
DeMorrow, Sharon
Published in
Cancer research (Chicago, Ill.)
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The anti‐glioblastoma drug ONC201 and related analogs act as non‐competitive antagonists at the D2 dopamine receptor through unique binding site interactions
by
Cuoco, Caroline Ann
,
Free, R. Benjamin
,
Willette, Blair
,
Lane, J. Robert
,
Allen, Joshua E.
,
Sibley, David R.
Published in
The FASEB journal
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The anti‐glioblastoma drug ONC201 and related analogs act as non‐competitive antagonists at the D 2 dopamine receptor through unique binding site interactions
by
Cuoco, Caroline Ann
,
Free, R. Benjamin
,
Willette, Blair
,
Lane, J. Robert
,
Allen, Joshua E.
,
Sibley, David R.
Published in
The FASEB journal
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DDRE-33. MOLECULAR DIFFERENTIATION OF IMIPRIDONES ONC201 AND ONC206
by
Prabhu, Varun
,
Cuoco, Caroline
,
Jung, Jinkyu
,
Morrow, Sara
,
Kawakibi, Abed Rahman
,
Willette, Blair
,
Day, Marilyn
,
Anantharaman, Lakshmi
,
Charter, Neil
,
Rucker, Joseph
,
Doranz, Benjamin
,
Basken, Joel
,
Stogniew, Martin
,
Gilbert, Mark
,
Free, R
,
Sibley, David
,
Allen, Joshua
Published in
Neuro-oncology (Charlottesville, Va.)
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Abstract A22: Molecular subtypes and resistance programs in pancreatic ductal adenocarcinoma elucidated with single-nucleus RNA-seq
by
Hwang, William L.
,
Jagadeesh, Karthik A.
,
Ashenberg, Orr
,
Drokhlyansky, Eugene
,
Eng, George
,
Wittenberghe, Nicholas Van
,
Freed-Pastor, William
,
Rodriguez, Clifton
,
Dionne, Danielle
,
Waldman, Julia
,
Cuoco, Michael
,
Tsankov, Alexander
,
Lambden, Connor
,
Porter, Caroline
,
Schenkel, Jason
,
Lambert, Laurens
,
Ciprani, Debora
,
Aguirre, Andrew J.
,
Mino-Kenudson, Mari
,
Hong, Theodore S.
,
Rozenblatt-Rosen, Orit
,
Castillo, Carlos Fernandez-del
,
Liss, Andrew S.
,
Regev, Aviv
,
Jacks, Tyler E.
Published in
Cancer research (Chicago, Ill.)
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DDIS-20. IMIPRIDONE STRUCTURE ACTIVITY RELATIONSHIP UNCOVERS ONC206 AS THE NEXT BITOPIC DRD2 ANTAGONIST FOR ONCOLOGY WITH DIFFERENTIATED RECEPTOR PHARMACOLOGY
by
Prabhu, Varun
,
Cuoco, Caroline
,
Jung, Jinkyu
,
Rahman Kawakibi, Abed
,
Willette, Blair
,
Day, Marilyn
,
Anantharaman, Lakshmi
,
Charter, Neil
,
Rucker, Joseph
,
Doranz, Benjamin
,
Oster, Wolfgang
,
Stogniew, Martin
,
Gilbert, Mark
,
Benjamin Free, R
,
Sibley, David
,
Allen, Joshua
Published in
Neuro-oncology (Charlottesville, Va.)
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EXTH-33. RECEPTOR PHARMACOLOGY OF ONC201: THE FIRST BITOPIC DRD2 ANTAGONIST FOR CLINICAL NEURO-ONCOLOGY
by
Benjamin Free, R
,
Cuoco, Caroline
,
Prabhu, Varun
,
Willette, Blair
,
Day, Marilyn
,
Anantharaman, Lakshmi
,
Sulli, Chidananda
,
Davidson, Edgar
,
Deacon, Sean
,
Rucker, Joseph
,
Charter, Neil
,
Doranz, Benjamin
,
Oster, Wolfgang
,
Stogniew, Martin
,
Robert Lane, J
,
Sibley, David
,
Allen, Joshua
Published in
Neuro-oncology (Charlottesville, Va.)
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