Oral bioavailability and multiple dose tolerability of an antisense oligonucleotide tablet formulated with sodium caprate by Raoof, Araz A., Chiu, Peter, Ramtoola, Zeibun, Cumming, Iain K., Teng, Chingleou, Weinbach, Susan P., Hardee, Greg E., Levin, Arthur A., Geary, R.S.

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Structure-Based Design of Potent and Selective Inhibitors of the Metabolic Kinase PFKFB3 by Boyd, Scott, Brookfield, Joanna L, Critchlow, Susan E, Cumming, Iain A, Curtis, Nicola J, Debreczeni, Judit, Degorce, Sébastien L, Donald, Craig, Evans, Nicola J, Groombridge, Sam, Hopcroft, Philip, Jones, Neil P, Kettle, Jason G, Lamont, Scott, Lewis, Hilary J, MacFaull, Philip, McLoughlin, Sheila B, Rigoreau, Laurent J. M, Smith, James M, St-Gallay, Steve, Stock, Julie K, Turnbull, Andrew P, Wheatley, Edward R, Winter, Jon, Wingfield, Jonathan

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Structure-Based Design and Pharmacokinetic Optimization of Covalent Allosteric Inhibitors of the Mutant GTPase KRASG12C by Kettle, Jason G, Bagal, Sharan K, Bickerton, Sue, Bodnarchuk, Michael S, Breed, Jason, Carbajo, Rodrigo J, Cassar, Doyle J, Chakraborty, Atanu, Cosulich, Sabina, Cumming, Iain, Davies, Michael, Eatherton, Andrew, Evans, Laura, Feron, Lyman, Fillery, Shaun, Gleave, Emma S, Goldberg, Frederick W, Harlfinger, Stephanie, Hanson, Lyndsey, Howard, Martin, Howells, Rachel, Jackson, Anne, Kemmitt, Paul, Kingston, Jennifer K, Lamont, Scott, Lewis, Hilary J, Li, Songlei, Liu, Libin, Ogg, Derek, Phillips, Christopher, Polanski, Radek, Robb, Graeme, Robinson, David, Ross, Sarah, Smith, James M, Tonge, Michael, Whiteley, Rebecca, Yang, Junsheng, Zhang, Longfei, Zhao, Xiliang

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Discovery of AZD4625, a Covalent Allosteric Inhibitor of the Mutant GTPase KRASG12C by Kettle, Jason G., Bagal, Sharan K., Bickerton, Sue, Bodnarchuk, Michael S., Boyd, Scott, Breed, Jason, Carbajo, Rodrigo J., Cassar, Doyle J., Chakraborty, Atanu, Cosulich, Sabina, Cumming, Iain, Davies, Michael, Davies, Nichola L., Eatherton, Andrew, Evans, Laura, Feron, Lyman, Fillery, Shaun, Gleave, Emma S., Goldberg, Frederick W., Hanson, Lyndsey, Harlfinger, Stephanie, Howard, Martin, Howells, Rachel, Jackson, Anne, Kemmitt, Paul, Lamont, Gillian, Lamont, Scott, Lewis, Hilary J., Liu, Libin, Niedbala, Michael J., Phillips, Christopher, Polanski, Radek, Raubo, Piotr, Robb, Graeme, Robinson, David M., Ross, Sarah, Sanders, Matthew G., Tonge, Michael, Whiteley, Rebecca, Wilkinson, Stephen, Yang, Junsheng, Zhang, Wenman

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Discovery of AZD4625, a Covalent Allosteric Inhibitor of the Mutant GTPase KRAS G12C by Kettle, Jason G, Bagal, Sharan K, Bickerton, Sue, Bodnarchuk, Michael S, Boyd, Scott, Breed, Jason, Carbajo, Rodrigo J, Cassar, Doyle J, Chakraborty, Atanu, Cosulich, Sabina, Cumming, Iain, Davies, Michael, Davies, Nichola L, Eatherton, Andrew, Evans, Laura, Feron, Lyman, Fillery, Shaun, Gleave, Emma S, Goldberg, Frederick W, Hanson, Lyndsey, Harlfinger, Stephanie, Howard, Martin, Howells, Rachel, Jackson, Anne, Kemmitt, Paul, Lamont, Gillian, Lamont, Scott, Lewis, Hilary J, Liu, Libin, Niedbala, Michael J, Phillips, Christopher, Polanski, Radek, Raubo, Piotr, Robb, Graeme, Robinson, David M, Ross, Sarah, Sanders, Matthew G, Tonge, Michael, Whiteley, Rebecca, Wilkinson, Stephen, Yang, Junsheng, Zhang, Wenman

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A novel series of positive modulators of the AMPA receptor: Discovery and structure based hit-to-lead studies by Jamieson, Craig, Basten, Stephanie, Campbell, Robert A., Cumming, Iain A., Gillen, Kevin J., Gillespie, Jonathan, Kazemier, Bert, Kiczun, Michael, Lamont, Yvonne, Lyons, Amanda J., Maclean, John K.F., Moir, Elizabeth M., Morrow, John A., Papakosta, Marianthi, Rankovic, Zoran, Smith, Lynn

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Structure-Based Design and Pharmacokinetic Optimization of Covalent Allosteric Inhibitors of the Mutant GTPase KRAS G12C by Kettle, Jason G, Bagal, Sharan K, Bickerton, Sue, Bodnarchuk, Michael S, Breed, Jason, Carbajo, Rodrigo J, Cassar, Doyle J, Chakraborty, Atanu, Cosulich, Sabina, Cumming, Iain, Davies, Michael, Eatherton, Andrew, Evans, Laura, Feron, Lyman, Fillery, Shaun, Gleave, Emma S, Goldberg, Frederick W, Harlfinger, Stephanie, Hanson, Lyndsey, Howard, Martin, Howells, Rachel, Jackson, Anne, Kemmitt, Paul, Kingston, Jennifer K, Lamont, Scott, Lewis, Hilary J, Li, Songlei, Liu, Libin, Ogg, Derek, Phillips, Christopher, Polanski, Radek, Robb, Graeme, Robinson, David, Ross, Sarah, Smith, James M, Tonge, Michael, Whiteley, Rebecca, Yang, Junsheng, Zhang, Longfei, Zhao, Xiliang

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A novel series of positive modulators of the AMPA receptor: Structure-based lead optimization by Jamieson, Craig, Campbell, Robert A., Cumming, Iain A., Gillen, Kevin J., Gillespie, Jonathan, Kazemier, Bert, Kiczun, Michael, Lamont, Yvonne, Lyons, Amanda J., Maclean, John K.F., Martin, Frederic, Moir, Elizabeth M., Morrow, John A., Pantling, John, Rankovic, Zoran, Smith, Lynn

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Genome-Wide Methylation Profiling in 229 Patients With Crohn’s Disease Requiring Intestinal Resection: Epigenetic Analysis of the Trial of Prevention of Post-operative Crohn’s Dise... by Ventham, Nicholas T., Kennedy, Nicholas A., Kalla, Rahul, Adams, Alex T., Noble, Alexandra, Ennis, Holly, Arnott, Ian, Cahill, Aiden, Smith, Malcolm, Ahmad, Tariq, Subramanian, Sreedhar, Travis, Simon, Morris, John, Hamlin, John, Dhar, Anjan, Nwokolo, Chuka, Creed, Tom, Bloom, Stuart, Yousif, Mohamed, Thomas, Linzi, Campbell, Simon, Lewis, Stephen J., Sebastian, Shaji, Sen, Sandip, Lal, Simon, Hawkey, Chris, Murray, Charles, Cummings, Fraser, Goh, Jason, Lindsay, James O., Arebi, Naila, Potts, Lindsay, McKinley, Aileen J., Thomson, John M., Todd, John A., Collie, Mhairi, Mowat, Ashley, Gaya, Daniel R., Winter, Jack, Naismith, Graham D., Keerie, Catriona, Lewis, Steff, Prescott, Robin J., Campbell, Harry, McGovern, Dermot P.B., Annese, Vito, Zoldoš, Vlatka, Permberton, Iain K., Wuhrer, Manfred, Kolarich, Daniel, Fernandes, Daryl L., Theorodorou, Evropi, Daniel I. Spencer, Victoria Merrick, Gardner, Richard A., Doran, Ray, Shubhakar, Archana, Boyapati, Ray, Rudan, Igor, Lionetti, Paolo, Akmačić, Irena Trbojević, Krištić, Jasminka, Vuč ković, Frano, Štambuk, Jerko, Novokmet, Mislav, Pučić-Baković, Maja, Gornik, Olga, Andriulli, Angelo, Cantoro, Laura, Sturniolo, Giancarlo, Fiorino, Gionata, Manetti, Natalia, Latiano, Anna, Kohn, Anna, D’Inca`, Renata, Danese, Silvio, Arnott, Ian D., Noble, Colin L., Lees, Charlie W., Shand, Alan G., Murphy, Lee, Gibson, Jude, Evenden, Louise, Wrobel, Nicola, Gilchrist, Tamara, Fawkes, Angie, Kammeijer, Guinevere S.M., Clerc, Florent, de Haan, Noortje, Vojta, Aleksandar, Samaržija, Ivana, Markulin, Dora, Klasić, Marija, Dobrinić, Paula, Aulchenko, Yurii, van den Heuve, Tim, Jonkers, Daisy, Pierik, Marieke, Mowat, Craig, Dunlop, Malcolm G., Satsangi, Jack

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Design, synthesis, and structure–activity relationships of indole-3-carboxamides as novel water soluble cannabinoid CB1 receptor agonists by Adam, Julia M., Cairns, Jim, Caulfield, Wilson, Cowley, Phillip, Cumming, Iain, Easson, Morag, Edwards, Darren, Ferguson, Morag, Goodwin, Richard, Jeremiah, Fiona, Kiyoi, Takao, Mistry, Ashvin, Moir, Elizabeth, Morphy, Richard, Tierney, Jason, York, Mark, Baker, James, Cottney, Jean E., Houghton, Andrea K., Westwood, Paul J., Walker, Glenn

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The influence of birth weight and genetic factors on lipid levels: a study in adult twins by Tuya, Chuluuntulga, Mutch, William J., Haggarty, Paul, Campbell, Doris M., Cumming, Alastair, Kelly, Kevin, Broom, Iain, McNeill, Geraldine

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Design, synthesis, and structure-activity relationships of indole-3-carboxamides as novel water soluble cannabinoid CB1 receptor agonistsElectronic supplementary information (ESI)... by Adam, Julia M, Cairns, Jim, Caulfield, Wilson, Cowley, Phillip, Cumming, Iain, Easson, Morag, Edwards, Darren, Ferguson, Morag, Goodwin, Richard, Jeremiah, Fiona, Kiyoi, Takao, Mistry, Ashvin, Moir, Elizabeth, Morphy, Richard, Tierney, Jason, York, Mark, Baker, James, Cottney, Jean E, Houghton, Andrea K, Westwood, Paul J, Walker, Glenn

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