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Search Results - Culshaw, Janet D.
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Imidazo[1,2-a]pyridines. Part 2: SAR and optimisation of a potent and selective class of cyclin-dependent kinase inhibitors
by
BYTH, Kate F
,
CULSHAW, Janet D
,
GREEN, Stephen
,
OAKES, Sandra E
,
THOMAS, Andrew P
Published in
Bioorganic & medicinal chemistry letters
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Synthesis of 3-Substituted 2-Aminopyridines via Displacement of 3-Fluoro-2-nitropyridine
by
Culshaw, Janet D.
,
Eden, Jonathan M.
,
Ford, Susannah J.
,
Hayter, Barry
,
Perkins, David R.
,
Pike, Kurt G.
Published in
Synlett
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Imidazo[1,2- a]pyridines: A potent and selective class of cyclin-Dependent kinase inhibitors identified through structure-Based hybridisation
by
Anderson, Malcolm
,
Beattie, John F.
,
Breault, Gloria A.
,
Breed, Jason
,
Byth, Kate F.
,
Culshaw, Janet D.
,
Ellston, Rebecca P.A.
,
Green, Stephen
,
Minshull, Claire A.
,
Norman, Richard A.
,
Pauptit, Richard A.
,
Stanway, Judith
,
Thomas, Andrew P.
,
Jewsbury, Philip J.
Published in
Bioorganic & medicinal chemistry letters
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Imidazo[1,2-b]pyridazines: a potent and selective class of cyclin-dependent kinase inhibitors
by
BYTH, Kate F
,
COOPER, Nicola
,
PANNIFER, Andrew
,
ROWSELL, Sian
,
STANWAY, Judith J
,
VALENTINE, Anna L
,
THOMAS, Andrew P
,
CULSHAW, Janet D
,
HEATON, David W
,
OAKES, Sandra E
,
MINSHULL, Claire A
,
NORMAN, Richard A
,
PAUPTIT, Richard A
,
TUCKER, Julie A
,
BREED, Jason
Published in
Bioorganic & medicinal chemistry letters
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Imidazoles: SAR and development of a potent class of cyclin-dependent kinase inhibitors
by
Anderson, Malcolm
,
Andrews, David M.
,
Barker, Andy J.
,
Brassington, Claire A.
,
Breed, Jason
,
Byth, Kate F.
,
Culshaw, Janet D.
,
Finlay, M. Raymond V.
,
Fisher, Eric
,
McMiken, Helen H.J.
,
Green, Clive P.
,
Heaton, Dave W.
,
Nash, Ian A.
,
Newcombe, Nicholas J.
,
Oakes, Sandra E.
,
Pauptit, Richard A.
,
Roberts, Andrew
,
Stanway, Judith J.
,
Thomas, Andrew P.
,
Tucker, Julie A.
,
Walker, Mike
,
Weir, Hazel M.
Published in
Bioorganic & medicinal chemistry
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Imidazo[1,2-a]pyridines: A potent and selective class of cyclin-dependent kinase inhibitors identified through structure-based hybridisation: Recent advances in the design of kinas...
by
ANDERSON, Malcolm
,
BEATTIE, John F
,
PAUPTIT, Richard A
,
STANWAY, Judith
,
THOMAS, Andrew P
,
JEWSBURY, Philip J
,
BREAULT, Gloria A
,
BREED, Jason
,
BYTH, Kate F
,
CULSHAW, Janet D
,
ELLSTON, Rebecca P. A
,
GREEN, Stephen
,
MINSHULL, Claire A
,
NORMAN, Richard A
Published in
Bioorganic & medicinal chemistry letters
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Correction to “Discovery of a Thiadiazole–Pyridazine-Based Allosteric Glutaminase 1 Inhibitor Series That Demonstrates Oral Bioavailability and Activity in Tumor Xenograft Models”...
by
Finlay, M. Raymond V.
,
Anderton, Mark
,
Bailey, Andrew
,
Boyd, Scott
,
Brookfield, Joanna
,
Cairnduff, Ceri
,
Charles, Mark
,
Cheasty, Anne
,
Critchlow, Susan E.
,
Culshaw, Janet
,
Debreczeni, Judit
,
Ekwuru, Tennyson
,
Hollingsworth, Ian
,
Jones, Neil
,
Leroux, Fred
,
Littleson, Mairi
,
McCarron, Hollie
,
McKelvie, Jennifer
,
Mooney, Lorraine
,
Nissink, J. Willem M.
,
Patel, Joe
,
Perkins, David
,
Powell, Steve
,
Quesada, Mar Jimenez
,
Raubo, Piotr
,
Sabin, Verity
,
Smith, James
,
Smith, Peter D.
,
Stark, Andrew
,
Ting, Attilla
,
Wang, Peng
,
Wilson, Zena
,
Winter-Holt, Jon J.
,
Wood, J. Matthew
,
Wrigley, Gail L.
,
Yu, Guoqing
,
Zhang, Peng
Published in
Journal of medicinal chemistry
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8
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Discovery of a Thiadiazole–Pyridazine-Based Allosteric Glutaminase 1 Inhibitor Series That Demonstrates Oral Bioavailability and Activity in Tumor Xenograft Models
by
Finlay, M. Raymond V
,
Anderton, Mark
,
Bailey, Andrew
,
Boyd, Scott
,
Brookfield, Joanna
,
Cairnduff, Ceri
,
Charles, Mark
,
Cheasty, Anne
,
Critchlow, Susan E
,
Culshaw, Janet
,
Ekwuru, Tennyson
,
Hollingsworth, Ian
,
Jones, Neil
,
Leroux, Fred
,
Littleson, Mairi
,
McCarron, Hollie
,
McKelvie, Jennifer
,
Mooney, Lorraine
,
Nissink, J. Willem M
,
Perkins, David
,
Powell, Steve
,
Quesada, Mar Jimenez
,
Raubo, Piotr
,
Sabin, Verity
,
Smith, James
,
Smith, Peter D
,
Stark, Andrew
,
Ting, Attilla
,
Wang, Peng
,
Wilson, Zena
,
Winter-Holt, Jon J
,
Wood, J. Matthew
,
Wrigley, Gail L
,
Yu, Guoqing
,
Zhang, Peng
Published in
Journal of medicinal chemistry
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Discovery and Optimization of Pyrrolopyrimidine Inhibitors of Interleukin‑1 Receptor Associated Kinase 4 (IRAK4) for the Treatment of Mutant MYD88L265P Diffuse Large B‑Cell Lymphom...
by
Scott, James S
,
Degorce, Sébastien L
,
Anjum, Rana
,
Culshaw, Janet
,
Davies, Robert D. M
,
Davies, Nichola L
,
Dillman, Keith S
,
Dowling, James E
,
Drew, Lisa
,
Ferguson, Andrew D
,
Groombridge, Sam D
,
Halsall, Christopher T
,
Hudson, Julian A
,
Lamont, Scott
,
Lindsay, Nicola A
,
Marden, Stacey K
,
Mayo, Michele F
,
Pease, J. Elizabeth
,
Perkins, David R
,
Pink, Jennifer H
,
Robb, Graeme R
,
Rosen, Alan
,
Shen, Minhui
,
McWhirter, Claire
,
Wu, Dedong
Published in
Journal of medicinal chemistry
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10
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Discovery and Optimization of Pyrrolopyrimidine Inhibitors of Interleukin-1 Receptor Associated Kinase 4 (IRAK4) for the Treatment of Mutant MYD88 L265P Diffuse Large B-Cell Lympho...
by
Scott, James S
,
Degorce, Sébastien L
,
Anjum, Rana
,
Culshaw, Janet
,
Davies, Robert D M
,
Davies, Nichola L
,
Dillman, Keith S
,
Dowling, James E
,
Drew, Lisa
,
Ferguson, Andrew D
,
Groombridge, Sam D
,
Halsall, Christopher T
,
Hudson, Julian A
,
Lamont, Scott
,
Lindsay, Nicola A
,
Marden, Stacey K
,
Mayo, Michele F
,
Pease, J Elizabeth
,
Perkins, David R
,
Pink, Jennifer H
,
Robb, Graeme R
,
Rosen, Alan
,
Shen, Minhui
,
McWhirter, Claire
,
Wu, Dedong
Published in
Journal of medicinal chemistry
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