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Search Results - Bleam, Maureen R.
Search Results - Bleam, Maureen R.
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Dabrafenib; preclinical characterization, increased efficacy when combined with trametinib, while BRAF/MEK tool combination reduced skin lesions
by
King, Alastair J
,
Arnone, Marc R
,
Bleam, Maureen R
,
Moss, Katherine G
,
Yang, Jingsong
,
Fedorowicz, Kelly E
,
Smitheman, Kimberly N
,
Erhardt, Joseph A
,
Hughes-Earle, Angela
,
Kane-Carson, Laurie S
,
Sinnamon, Robert H
,
Qi, Hongwei
,
Rheault, Tara R
,
Uehling, David E
,
Laquerre, Sylvie G
Published in
PloS one
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Distinct Concentration-Dependent Effects of the Polo-like Kinase 1―Specific Inhibitor GSK461364A, Including Differential Effect on Apoptosis
by
GILMARTIN, Aidan G
,
BLEAM, Maureen R
,
SUTTON, David
,
DIAMOND, Melody A
,
JACKSON, Jeffrey R
,
LAQUERRE, Sylvie G
,
RICHTER, Mark C
,
ERSKINE, Symon G
,
KRUGER, Ryan G
,
MADDEN, Lenore
,
HASSLER, Daniel F
,
SMITH, Gary K
,
GONTAREK, Richard R
,
COURTNEY, Mary P
Published in
Cancer research (Chicago, Ill.)
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GSK1120212 (JTP-74057) Is an Inhibitor of MEK Activity and Activation with Favorable Pharmacokinetic Properties for Sustained In Vivo Pathway Inhibition
by
GILMARTIN, Aidan G
,
BLEAM, Maureen R
,
ZAPPACOSTA, Francesca
,
ANNAN, Roland
,
SUTTON, David
,
LAQUERRE, Sylvie G
,
GROY, Arthur
,
MOSS, Katherine G
,
MINTHORN, Elisabeth A
,
KULKARNI, Swarupa G
,
ROMINGER, Cynthia M
,
ERSKINE, Symon
,
FISHER, Kelly E
,
JINGSONG YANG
Published in
Clinical cancer research
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Combinations of BRAF, MEK, and PI3K/mTOR inhibitors overcome acquired resistance to the BRAF inhibitor GSK2118436 dabrafenib, mediated by NRAS or MEK mutations
by
Greger, James G
,
Eastman, Stephen D
,
Zhang, Vivian
,
Bleam, Maureen R
,
Hughes, Ashley M
,
Smitheman, Kimberly N
,
Dickerson, Scott H
,
Laquerre, Sylvie G
,
Liu, Li
,
Gilmer, Tona M
Published in
Molecular cancer therapeutics
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Abstract 2867: Inhibition of BET bromodomain proteins as a therapeutic approach in small cell lung cancer
by
Wyce, Anastasia
,
Le, BaoChau
,
Bai, Yuchen
,
Soong, David
,
Zhang, Xi-Ping
,
Matteo, Jeanne J.
,
Korenchuk, Susan
,
Butticello, Michael F.
,
Plant, Ramona
,
Bleam, Maureen R.
,
Degenhardt, Yan
,
McHugh, Charles F.
,
Carpenter, Christopher
,
Tummino, Peter J.
,
Barbash, Olena
Published in
Cancer research (Chicago, Ill.)
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Abstract B71: Acquired resistance to the BRAF inhibitor GSK2118436, mediated by NRAS or MEK mutation, can be overcome with combinations that inhibit BRAF and MEK, BRAF and PI3K/mTO...
by
Greger, James G.
,
Eastman, Stephen D.
,
Zhang, Vivian
,
Bleam, Maureen R.
,
Hughes, Ashley
,
Smitheman, Kimberly N.
,
Laquerre, Sylvie
,
Liu, Li
,
Gilmer, Tona M.
Published in
Molecular cancer therapeutics
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Janus Kinase (JAK) 1 Inhibition Results in Significant Changes in Serum Proteins and Peripheral T-Cell Populations That Correlated with Clinical Scores in Chronic Graft Versus Host...
by
Pratta, Michael
,
Volkova, Angelina
,
Bleam, Maureen
,
Morariu-Zamfir, Rodica
,
Rumberger, Beth
,
Douglass, Stephen
,
Smith, Susan H.
,
Bhatt, Valkal
,
Galvin, John
,
Im, Annie
,
Paczesny, Sophie
,
Schultz, Kirk R.
,
Pavletic, Steven Z.
Published in
Blood
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Janus Kinase (JAK) 1 Inhibition Results in Significant Changes in Serum Proteins and Peripheral T-Cell Populations That Correlate with Clinical Scores in Patients with Chronic Graf...
by
Pratta, Michael
,
Volkova, Angelina
,
Bleam, Maureen
,
Morariu-Zamfir, Rodica
,
Rumberger, Beth
,
Douglass, Stephen
,
Smith, Susan H.
,
Bhatt, Valkal
,
Galvin, John
,
Im, Dr. Annie
,
Paczesny, Sophie
,
Schultz, Kirk R.
,
Pavletic, Dr. Steven Z.
Published in
Transplantation and cellular therapy
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Identification and characterization of potent small molecule inhibitor of hemorrhagic fever New World arenaviruses
by
Bolken, Tove′ C.
,
Laquerre, Sylvie
,
Zhang, Yuanming
,
Bailey, Thomas R.
,
Pevear, Daniel C.
,
Kickner, Shirley S.
,
Sperzel, Lindsey E.
,
Jones, Kevin F.
,
Warren, Travis K.
,
Amanda Lund, S.
,
Kirkwood-Watts, Dana L.
,
King, David S.
,
Shurtleff, Amy C.
,
Guttieri, Mary C.
,
Deng, Yijun
,
Bleam, Maureen
,
Hruby, Dennis E.
Published in
Antiviral research
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