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N-Hydroxyformamide peptidomimetics as TACE/Matrix metalloprotease inhibitors: oral activity via P1′ isobutyl substitution
by
Musso, David L.
,
Andersen, Marc W.
,
Andrews, Robert C.
,
Austin, Richard
,
Beaudet, Elizabeth J.
,
Becherer, J.David
,
Bubacz, Dulce G.
,
Bickett, D.Mark
,
Chan, Joseph H.
,
Conway, James G.
,
Cowan, David J.
,
Gaul, Michael D.
,
Glennon, Kimberly C.
,
Hedeen, Kevin M.
,
Lambert, Millard H.
,
Leesnitzer, M.Anthony
,
McDougald, Darryl L.
,
Mitchell, Justin L.
,
Moss, Marcia L.
,
Rabinowitz, Michael H.
,
Rizzolio, Michele C.
,
Schaller, Lee T.
,
Stanford, Jennifer B.
,
Tippin, Timothy K.
,
Warner, Janet R.
,
Whitesell, L.Graham
,
Wiethe, Robert W.
Published in
Bioorganic & medicinal chemistry letters
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Bioorganic & Medicinal Chemistry Letters
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