Discovery, SAR, and X‑ray Binding Mode Study of BCATm Inhibitors from a Novel DNA-Encoded Library by Deng, Hongfeng, Zhou, Jingye, Sundersingh, Flora S, Summerfield, Jennifer, Somers, Don, Messer, Jeffrey A, Satz, Alexander L, Ancellin, Nicolas, Arico-Muendel, Christopher C, (Sargent) Bedard, Katie L, Beljean, Arthur, Belyanskaya, Svetlana L, Bingham, Ryan, Smith, Sarah E, Boursier, Eric, Carter, Paul, Centrella, Paolo A, Clark, Matthew A, Chung, Chun-wa, Davie, Christopher P, Delorey, Jennifer L, Ding, Yun, Franklin, G. Joseph, Grady, LaShadric C, Herry, Kenny, Hobbs, Clare, Kollmann, Christopher S, Morgan, Barry A, (Pothier) Kaushansky, Laura J, Zhou, Quan

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Discovery of Highly Potent and Selective Small Molecule ADAMTS‑5 Inhibitors That Inhibit Human Cartilage Degradation via Encoded Library Technology (ELT) by Deng, Hongfeng, O’Keefe, Heather, Davie, Christopher P, Lind, Kenneth E, Acharya, Raksha A, Franklin, G. Joseph, Larkin, Jonathan, Matico, Rosalie, Neeb, Michael, Thompson, Monique M, Lohr, Thomas, Gross, Jeffrey W, Centrella, Paolo A, O’Donovan, Gary K, Bedard, Katie L. (Sargent), van Vloten, Kurt, Mataruse, Sibongile, Skinner, Steven R, Belyanskaya, Svetlana L, Carpenter, Tiffany Y, Shearer, Todd W, Clark, Matthew A, Cuozzo, John W, Arico-Muendel, Christopher C, Morgan, Barry A

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